SCHEMBL5072231

SCHEMBL5072231

O=C(O)NC1CCN(CC(=O)c2ccccc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 1/20 0.58
ADRA1A P35348 1/20 0.58
ADRA1B P35368 1/20 0.58
ALDH1A1 P00352 2/20 0.57
CARM1 Q86X55 1/20 0.53
PRMT6 Q96LA8 1/20 0.53
HTR2A P28223 1/20 0.52
HTR2C P28335 1/20 0.52
KCNH2 Q12809 1/20 0.52
KMT2A Q03164 2/20 0.52
MEN1 O00255 1/20 0.52
DRD4 P21917 1/20 0.51
MCHR1 Q99705 1/20 0.50
EPHX1 P07099 1/20 0.50
POLB P06746 1/20 0.50
SIGMAR1 Q99720 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21748573 0.87 ALDH1A1 (0.57) ALDH1A1KMT2AMEN1DRD4MCHR1
SCHEMBL13857680 0.82 KCNA3 (0.60) ADRA1DADRA1AADRA1BALDH1A1CARM1
SCHEMBL12424250 0.80 ALDH1A1 (0.56) ALDH1A1HTR2AHTR2CKCNH2KMT2A
SCHEMBL4875267 0.80 ALDH1A1 (0.79) ALDH1A1HTR2AHTR2CKCNH2KMT2A
SCHEMBL12859265 0.80 KMT2A (0.64) ALDH1A1HTR2AHTR2CKCNH2KMT2A
SCHEMBL14189783 0.80 ALDH1A1 (0.59) ALDH1A1HTR2AHTR2CKCNH2KMT2A
SCHEMBL4308106 0.80 ALDH1A1 (0.59) ALDH1A1HTR2AHTR2CKCNH2KMT2A
SCHEMBL9500234 0.78 HTR2A (0.64) ALDH1A1HTR2AHTR2CKCNH2KMT2A
SCHEMBL2425554 0.78 SIGMAR1 (0.78) KMT2ADRD4MCHR1POLBSIGMAR1
SCHEMBL6232219 0.77 ALDH1A1 (0.56) ALDH1A1HTR2AHTR2CKCNH2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874318-A2 N-ALKYL-AZACYCLOALKYL NMDA/NR2B ANTAGONISTS Merck & Co., Inc. (US) 2008-01-09 EP disclosed
WO-2006113471-A2 N-ALKYL-AZACYCLOALKYL NMDA/NR2B ANTAGONISTS MERCK & CO., INC. (US) 2006-10-26 WO disclosed