SCHEMBL5074359

SCHEMBL5074359

C[C](Cc1ccccc1)C(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.48
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
AKR1B1 P15121 1/20 0.46
TRPA1 O75762 2/20 0.43
TAAR1 Q96RJ0 3/20 0.43
SLC6A2 P23975 2/20 0.43
MAOA P21397 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
CYP2A6 P11509 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
POLB P06746 1/20 0.42
CNR2 P34972 2/20 0.41
TP53 P04637 1/20 0.40
SLC18A2 Q05940 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9513104 0.84 CES2 (0.50) TSHRCES2CES1AKR1B1TRPA1
SCHEMBL7369705 0.78 TSHR (0.50) TSHRCES2CES1AKR1B1TRPA1
SCHEMBL3245857 0.78 TSHR (0.50) TSHRCES2CES1AKR1B1TRPA1
SCHEMBL22338912 0.77 TSHR (0.50) TSHRCES2CES1AKR1B1TRPA1
SCHEMBL8105873 0.77 TRPA1 (0.50) TSHRTRPA1TAAR1SLC6A2MAOA
SCHEMBL8106172 0.77 MEN1 (0.43) TSHRCES2CES1AKR1B1TRPA1
SCHEMBL6616395 0.76 TSHR (0.44) TSHRCES2CES1AKR1B1CNR2
SCHEMBL11339635 0.75 CES1 (0.50) TSHRCES2CES1AKR1B1TP53
SCHEMBL531194 0.75 CES1 (0.50) TSHRCES2CES1AKR1B1TP53
Benzene SCHEMBL9806260 0.75 CES1 (0.50) TSHRCES2CES1AKR1B1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4118948-B2 2008-07-16 JP claimed
EP-0861026-B1 SYNERGISTIC HERBICIDAL MIXTURES CONTAINING CYCLOHEXENONE OXIME ETHER BASF AG (DE) 2003-04-02 EP claimed
JP-2000503297-A 2000-03-21 JP claimed
EP-0861026-A1 SYNERGISTIC HERBICIDAL MIXTURES CONTAINING CYCLOHEXENONE OXIME ETHER BASF AKTIENGESELLSCHAFT (DE) 1998-09-02 EP claimed
WO-1997010710-A1 SYNERGISTIC HERBICIDAL MIXTURES CONTAINING CYCLOHEXENONE OXIME ETHER BASF AKTIENGESELLSCHAFT (DE) 1997-03-27 WO claimed
WO-2016087593-A1 NOVEL FUNGICIDAL QUINOLINYLAMIDINES SYNGENTA PARTICIPATIONS AG (CH) 2016-06-09 WO disclosed
WO-2006078275-A2 IONIC LIQUID ENERGETIC MATERIALS LIOTTA CHARLES L (US) 2006-07-27 WO disclosed
CN-1312680-A Herbicidal compositions containing acylated aminophenylsulfonylureas AVENTIES CROP SCIENCES GMBH (DE) 2001-09-12 CN disclosed
WO-1999031988-A1 PLANT GROWTH REGULATION CELGENE CORPORATION (US) 1999-07-01 WO disclosed
US-5866512-A CONTROLLING WEEDS CELGENE CORPORATION (US) 1999-02-02 US disclosed
EP-0871609-A1 CYCLOHEXENONE OXIME ETHER METAL SALTS BASF AKTIENGESELLSCHAFT (DE) 1998-10-21 EP disclosed
EP-0861026-A1 SYNERGISTIC HERBICIDAL MIXTURES CONTAINING CYCLOHEXENONE OXIME ETHER BASF AKTIENGESELLSCHAFT (DE) 1998-09-02 EP disclosed
WO-1997020807-A1 CYCLOHEXENONE OXIME ETHER METAL SALTS BASF AKTIENGESELLSCHAFT (DE) 1997-06-12 WO disclosed
WO-1997010710-A1 SYNERGISTIC HERBICIDAL MIXTURES CONTAINING CYCLOHEXENONE OXIME ETHER BASF AKTIENGESELLSCHAFT (DE) 1997-03-27 WO disclosed