SCHEMBL5074496

SCHEMBL5074496

O=C(O)N1CCN(C2CNC2)C(CO)C1

nearest known ligand 0.31

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.31
CHRNB4 P30926 2/20 0.31
CHRNA3 P32297 2/20 0.31
CHRNA4 P43681 2/20 0.31
CHRNA7 P36544 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3225291 0.88 LMNA (0.37)
SCHEMBL694082 0.81 CHRNB2 (0.52) CHRNB2CHRNB4CHRNA3CHRNA4CHRNA7
SCHEMBL3225724 0.79 NR1H2 (0.45)
SCHEMBL4878901 0.77 POLB (0.34)
SCHEMBL4664823 0.77 POLB (0.34)
SCHEMBL16093727 0.75 CHRNB2 (0.32) CHRNB2CHRNB4CHRNA3CHRNA4CHRNA7
SCHEMBL4630301 0.74 POLB (0.40)
SCHEMBL17621805 0.74 OPRK1 (0.30)
SCHEMBL22530795 0.72 CHRNB2 (0.34) CHRNB2CHRNB4CHRNA3CHRNA4CHRNA7
SCHEMBL22530366 0.72 CHRNB2 (0.34) CHRNB2CHRNB4CHRNA3CHRNA4CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899326-A1 NEW AZETIDINE DERIVATIVES AS NEUROKININ RECEPTOR ANTAGONISTS FOR THE TREATMENT OF GASTROINTESTINAL DISEASES AstraZeneca AB (SE) 2008-03-19 EP disclosed
WO-2006137790-A1 NEW AZETIDINE DERIVATIVES AS NEUROKININ RECEPTOR ANTAGONISTS FOR THE TREATMENT OF GASTROINTESTINAL DISEASES ASTRAZENECA AB (SE) 2006-12-28 WO disclosed