SCHEMBL5078717

SCHEMBL5078717

FC(F)(F)c1ncc(-c2ccccc2)cn1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
NPC1 O15118 2/20 0.54
NFKB1 P19838 2/20 0.54
NFKB2 Q00653 2/20 0.54
RELA Q04206 2/20 0.54
KIF11 P52732 1/20 0.48
ATM Q13315 1/20 0.44
ALDH1A1 P00352 3/20 0.41
DHFR P00374 1/20 0.40
SCN2A Q99250 3/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39
CCNE2 O96020 1/20 0.37
CDK4 P11802 1/20 0.37
CCND1 P24385 1/20 0.37
CCNE1 P24864 1/20 0.37
CDK2 P24941 1/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Biphenyl SCHEMBL27729747 0.84 KIF11 (0.50) RAB9ASMN1; SMN2NPC1NFKB1NFKB2
SCHEMBL24155913 0.79 RAB9A (0.58) RAB9ASMN1; SMN2NPC1ALDH1A1L3MBTL1
SCHEMBL26635446 0.78 NPC1 (0.44) RAB9ASMN1; SMN2NPC1ALDH1A1L3MBTL1
SCHEMBL31375503 0.78 NPSR1 (0.42) RAB9ASMN1; SMN2NPC1NFKB1NFKB2
SCHEMBL18101370 0.77 RAB9A (0.54) RAB9ASMN1; SMN2NPC1NFKB1NFKB2
Biphenyl SCHEMBL27928291 0.77 GAA (0.42) RAB9ANPC1KIF11ALDH1A1MAPT
SCHEMBL16906666 0.77 AR (0.46) RAB9ASMN1; SMN2NPC1ATMALDH1A1
SCHEMBL17619727 0.75 CYP2A6 (0.48) RAB9ASMN1; SMN2NPC1ALDH1A1L3MBTL1
SCHEMBL16404616 0.74 TRPV4 (0.52) RAB9ASMN1; SMN2NPC1NFKB1NFKB2
SCHEMBL16903671 0.74 KIF11 (0.53) KIF11ATMALDH1A1DHFRSCN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1973884-A2 NOVEL HETEROCYCLES Orchid Research Laboratories Limited (IN) 2008-10-01 EP claimed
WO-2007083182-A2 NOVEL HETEROCYCLES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-07-26 WO claimed
CN-116621778-A USP inhibitor, preparation method and application thereof 北京华森英诺生物科技有限公司 2023-08-22 CN disclosed
CN-109476640-B Bicyclic proline compounds 豪夫迈·罗氏有限公司 2022-02-25 CN disclosed
CN-101360717-A Novel heterocycles ORCHID RES LAB LTD (IN) 2009-02-04 CN disclosed