SCHEMBL5082342

SCHEMBL5082342

CN1CCN(Cc2cc(C=CC(=O)N(C)Cc3cc4ccccc4o3)cnc2N)CC1

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.40
HTR2B P41595 3/20 0.40
DRD2 P14416 2/20 0.40
HRH3 Q9Y5N1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5082332 1.00 HTR1A (0.40) HTR1AHTR2BDRD2HRH3
Hydrochloric Acid SCHEMBL1253093 0.99 HTR1A (0.39) HTR1AHTR2BDRD2HRH3
Hydrochloric Acid SCHEMBL1253096 0.99 HTR1A (0.39) HTR1AHTR2BDRD2HRH3
SCHEMBL5082745 0.83 FAAH (0.39)
SCHEMBL5082771 0.83 FAAH (0.39)
Hydrochloric Acid SCHEMBL1254161 0.82 FAAH (0.39)
Hydrochloric Acid SCHEMBL1254167 0.82 FAAH (0.39)
SCHEMBL5076267 0.80 KIT (0.41)
Hydrochloric Acid SCHEMBL1251761 0.79 KIT (0.40)
Hydrochloric Acid SCHEMBL1251765 0.79 KIT (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1608377-B1 PHARMACEUTICAL COMPOSITIONS COMPRISING INHIBITORS OF FAB I AND FURTHER ANTIBIOTICS AFFINIUM PHARM INC (CA) 2008-10-01 EP claimed