SCHEMBL5082457

SCHEMBL5082457

CCN(CC)c1ncnc2c1ncn2C(CO)CCOCP(=O)(O)OC(OC(=O)OC(C)C)OC(=O)OC(C)C

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 3/20 0.38
FAP Q12884 2/20 0.33
CYP3A4 P08684 4/20 0.31
CYP2D6 P10635 4/20 0.31
RGS12 O14924 1/20 0.31
CYP2C9 P11712 1/20 0.31
GNAI1 P63096 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
ALOX15 P16050 1/20 0.31
KMT2A Q03164 1/20 0.31
ENTPD3 O75355 1/20 0.31
NT5E P21589 1/20 0.31
ENPP1 P22413 1/20 0.31
ENTPD1 P49961 1/20 0.31
SLC22A6 Q4U2R8 1/20 0.31
AHCY P23526 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5082361 0.88 FGFR1 (0.47) FGFR1FAPCYP3A4CYP2D6SLC22A6
SCHEMBL5083025 0.83 POLB (0.38) FGFR1CYP3A4CYP2D6CYP1A2
SCHEMBL5082979 0.82 DNPH1 (0.37) FGFR1CYP1A2
SCHEMBL5086107 0.82 FGFR1 (0.37) FGFR1CYP3A4CYP2D6CYP1A2
SCHEMBL5080065 0.81 FGFR1 (0.44) FGFR1FAPCYP3A4CYP2D6ENPP1
SCHEMBL5082976 0.81 FAP (0.43) FGFR1FAPCYP3A4CYP2D6SLC22A6
SCHEMBL6689879 0.75 FGFR1 (0.41) FGFR1CYP3A4SLC22A6AHCY
SCHEMBL6696336 0.75 FGFR1 (0.43) FGFR1CYP3A4CYP2D6CYP1A2SLC22A6
SCHEMBL5082281 0.71 FGFR1 (0.46) FGFR1FAPCYP3A4CYP2D6ENPP1
SCHEMBL6316076 0.70 FGFR1 (0.61) FGFR1CYP3A4ENPP1SLC22A6AHCY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7388002-B2 Nucleosides, preparation thereof and use as inhibitors of RNA viral polymerases BIOCRYST PHARMACEUTICALS, INC. (US) 2008-06-17 US disclosed
US-20060122391-A1 Nucleosides, preparation thereof and use as inhibitors of RNA viral polymerases BIOCRYST PHARMACEUTICALS, INC. (US) 2006-06-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060122391-A1 Nucleosides, preparation thereof and use as inhibitors of RNA viral polymerases POLR2H, NSUN2, POLR2E FGFR1 3600/4885FAP 4556/4885CYP3A4 941/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.