SCHEMBL5082690

SCHEMBL5082690

COS(=O)(=O)c1cccc([N+](=O)[O-])c1[C@@]1(C)CO1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.41
MEN1 O00255 4/20 0.41
F2 P00734 1/20 0.39
PRSS1 P07477 1/20 0.39
PRSS2 P07478 1/20 0.39
PRSS3 P35030 1/20 0.39
THRB P10828 1/20 0.37
TDP1 Q9NUW8 3/20 0.37
POLB P06746 3/20 0.37
PKM P14618 2/20 0.37
ATM Q13315 1/20 0.37
ALDH1A1 P00352 4/20 0.36
HPGD P15428 2/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36
MMP8 P22894 1/20 0.36
MMP13 P45452 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1317710 0.76 KMT2A (0.63) KMT2AMEN1F2PRSS1PRSS2
SCHEMBL29508624 0.76 KMT2A (0.63) KMT2AMEN1F2PRSS1PRSS2
SCHEMBL10482176 0.75 TDP1 (0.58) KMT2AMEN1F2PRSS1PRSS2
SCHEMBL10654745 0.75 KMT2A (0.49) KMT2AMEN1F2PRSS1PRSS2
SCHEMBL6255181 0.72 TDP1 (0.46) KMT2AMEN1F2PRSS1PRSS2
SCHEMBL11817089 0.66 ALDH1A1 (0.52) KMT2AMEN1TDP1ALDH1A1HPGD
SCHEMBL29474818 0.66 KMT2A (0.58) KMT2AMEN1F2PRSS1PRSS2
SCHEMBL1953366 0.66 KMT2A (0.39) KMT2AMEN1F2PRSS1PRSS2
SCHEMBL3282597 0.66 KMT2A (0.39) KMT2AMEN1F2PRSS1PRSS2
SCHEMBL1953369 0.66 KMT2A (0.39) KMT2AMEN1F2PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008096136-A1 COMBINATIONS WITH A MUSCARINIC RECEPTOR ANTAGONIST ARGENTA DISCOVERY LTD (GB) 2008-08-14 WO disclosed
EP-1521757-A1 NOVEL TRICYCLIC SPIROPIPERIDINES OR SPIROPYRROLIDINES AstraZeneca AB (SE) 2005-04-13 EP disclosed
WO-2004005295-A1 NOVEL TRICYCLIC SPIROPIPERIDINES OR SPIROPYRROLIDINES ASTRAZENECA AB (SE) 2004-01-15 WO disclosed