Testolactone

Testolactone

SCHEMBL5083091

C[C@]12C=CC(=O)C=C1CC[C@@H]1[C@@H]2CC[C@]2(C)OC(=O)CC[C@@H]12.O=P(O)(O)O

nearest known ligand 0.89

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CYP19A1

The experimentally established mechanism targets of Testolactone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP19A1 known ✓ P11511 15/20 0.89
LMNA P02545 2/20 0.89
MAPT P10636 2/20 0.89
CYP3A4 P08684 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Testolactone SCHEMBL2300061 0.94 CYP19A1 (1.00) CYP19A1LMNAMAPTCYP3A4
Testolactone SCHEMBL4053 0.94 CYP19A1 (1.00) CYP19A1LMNAMAPTCYP3A4
SCHEMBL8980363 0.79 CYP19A1 (0.72) CYP19A1LMNAMAPTCYP3A4
SCHEMBL23691780 0.78 CYP19A1 (0.67) CYP19A1LMNAMAPTCYP3A4
SCHEMBL8393653 0.76 CYP19A1 (0.67) CYP19A1LMNAMAPTCYP3A4
Androstenedone SCHEMBL14450072 0.75 CYP19A1 (1.00) CYP19A1LMNAMAPTCYP3A4
Androstenedone SCHEMBL3758714 0.75 CYP19A1 (1.00) CYP19A1LMNAMAPTCYP3A4
Androstenedone SCHEMBL1144460 0.75 CYP19A1 (1.00) CYP19A1LMNAMAPTCYP3A4
Androstenedone SCHEMBL134061 0.75 CYP19A1 (1.00) CYP19A1LMNAMAPTCYP3A4
Androstenedone SCHEMBL12430773 0.75 CYP19A1 (1.00) CYP19A1LMNAMAPTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080044390-A1 Methods and compositions for the treatment of neurodegenerative disorders CHDI, INCORPORATED 2008-02-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080044390-A1 Methods and compositions for the treatment of neurodegenerative disorders HTT, SNCA, NLN CYP19A1 3938/4885LMNA 415/4885MAPT 9/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.