SCHEMBL5085838

SCHEMBL5085838

CCN(CC)C(=O)c1cc(OC)c2c(c1)C(=O)c1cccc(OC)c1C2=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.52
HPGD P15428 3/20 0.50
HSP90AA1 P07900 2/20 0.50
HSP90AB1 P08238 2/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
ALDH1A1 P00352 2/20 0.50
TTR P02766 2/20 0.50
LMNA P02545 2/20 0.50
CYP1A2 P05177 1/20 0.50
BLM P54132 1/20 0.50
KDM4E B2RXH2 1/20 0.50
ABCC4 O15439 1/20 0.50
USP2 O75604 1/20 0.50
TP53 P04637 1/20 0.50
CHRM2 P08172 1/20 0.50
HTR1A P08908 1/20 0.50
ADRA2A P08913 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
MAPT P10636 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8996333 0.86 MEN1 (0.53) HPGDHSP90AA1HSP90AB1MEN1KMT2A
SCHEMBL8996312 0.82 TTR (0.71) HPGDHSP90AA1HSP90AB1MEN1KMT2A
SCHEMBL5088188 0.81 CYP1A2 (0.48) KEAP1HPGDHSP90AA1HSP90AB1MEN1
SCHEMBL8996338 0.81 MEN1 (0.55) HPGDHSP90AA1HSP90AB1MEN1KMT2A
SCHEMBL8996342 0.79 ELANE (0.49) HPGDHSP90AA1HSP90AB1MEN1KMT2A
SCHEMBL26187353 0.75 TTR (0.54) KEAP1MEN1KMT2AALDH1A1TTR
SCHEMBL30609982 0.75 TTR (0.54) KEAP1MEN1KMT2AALDH1A1TTR
SCHEMBL9877831 0.75 HTR1A (0.50) MEN1KMT2AALDH1A1CYP1A2HTR1A
SCHEMBL8947495 0.75 EGFR (0.73) MEN1KMT2AALDH1A1LMNAKDM4E
SCHEMBL15413441 0.75 MEN1 (0.49) HPGDHSP90AA1HSP90AB1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008090078-A1 METHOD FOR THE SYNTHESIS OF RHEIN AND DERIVATIVES THEREOF PIERRE FABRE MEDICAMENT (FR) 2008-07-31 WO disclosed