SCHEMBL5086741

SCHEMBL5086741

NC(=O)Nc1c(CCCCN2CCN(c3ccc4c(c3)OCCO4)CC2)sc2ccccc12.NC(=O)Nc1cn(CCCCN2CCN(c3ccc4c(c3)OCO4)CC2)c2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 2/20 0.47
ADRA2A P08913 1/20 0.47
ADRA2B P18089 1/20 0.47
ADRA2C P18825 1/20 0.47
ADRA1A P35348 1/20 0.47
ADRA1B P35368 1/20 0.47
HTR1A P08908 5/20 0.45
SLC6A4 P31645 1/20 0.39
IGF2BP1 Q9NZI8 1/20 0.39
CNR2 P34972 1/20 0.38
MAPT P10636 1/20 0.37
OPRK1 P41145 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5088798 0.95 HTR1A (0.43) ADRA1DADRA2AADRA2BADRA2CADRA1A
SCHEMBL4950602 0.90 ADRA2A (0.53) ADRA1DADRA2AADRA2BADRA2CADRA1A
SCHEMBL4950289 0.90 HTR1A (0.52) ADRA1DADRA2AADRA2BADRA2CADRA1A
SCHEMBL4948057 0.87 HTR1A (0.49) ADRA1DADRA2AADRA2BADRA2CADRA1A
SCHEMBL4949840 0.87 HTR1A (0.49) ADRA1DADRA2AADRA2BADRA2CADRA1A
SCHEMBL4949561 0.87 ADRA1D (0.52) ADRA1DADRA2AADRA2BADRA2CADRA1A
SCHEMBL4950504 0.87 HTR1A (0.51) ADRA1DADRA2AADRA2BADRA2CADRA1A
SCHEMBL4945095 0.84 HTR1A (0.48) ADRA1DADRA2AADRA2BADRA2CADRA1A
SCHEMBL4950861 0.84 HTR1A (0.47) ADRA1DADRA2AADRA2BADRA2CADRA1A
SCHEMBL4948056 0.82 HTR1A (0.43) ADRA1DADRA2AADRA2BADRA2CADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2008526700-A 2008-07-24 JP claimed
EP-1761524-A1 PHENYL DIAZEPANE CARBOXAMIDES AND ANNELATED PHENYL PIPERAZINE CARBOXAMIDES CONTAINING OXYGEN AND USED AS DOPAMINE D3 ANTAGONISTS SCHWARZ PHARMA AG (DE) 2007-03-14 EP claimed
WO-2006072430-A1 PHENYL DIAZEPANE CARBOXAMIDES AND ANNELATED PHENYL PIPERAZINE CARBOXAMIDES CONTAINING OXYGEN AND USED AS DOPAMINE D3 ANTAGONISTS SCHWARZ PHARMA AG (DE) 2006-07-13 WO claimed