SCHEMBL5095709

SCHEMBL5095709

NC(=O)Nc1c(CCCCN2CCN(c3ccc4c(c3)OCCCO4)CC2)oc2ccccc12.NC(=O)Nc1cn(CCCCN2CCN(c3ccc4c(c3)OCCCO4)CC2)c2ccccc12

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.43
ADRA1D P25100 3/20 0.41
ADRA1A P35348 2/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
ADRA1B P35368 1/20 0.41
SLC6A4 P31645 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.36
CNR2 P34972 1/20 0.36
IGF2BP1 Q9NZI8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4949448 0.92 HTR1A (0.49) HTR1AADRA1DADRA1AADRA2AADRA2B
SCHEMBL4950861 0.90 HTR1A (0.47) HTR1AADRA1DADRA1AADRA2AADRA2B
SCHEMBL4950306 0.89 HTR1A (0.50) HTR1AADRA1DADRA1AADRA2AADRA2B
SCHEMBL4952024 0.89 HTR1A (0.53) HTR1AADRA1DADRA1AADRA2AADRA2B
SCHEMBL4945095 0.86 HTR1A (0.48) HTR1AADRA1DADRA1AADRA2AADRA2B
SCHEMBL4950504 0.86 HTR1A (0.51) HTR1AADRA1DADRA1AADRA2AADRA2B
SCHEMBL4949703 0.86 ADRA2A (0.52) HTR1AADRA1DADRA1AADRA2AADRA2B
SCHEMBL4950975 0.84 HTR1A (0.42) HTR1AADRA1DADRA1AADRA2AADRA2B
SCHEMBL4950555 0.84 HTR1A (0.42) HTR1AADRA1DADRA1AADRA2AADRA2B
SCHEMBL4949561 0.83 ADRA1D (0.52) HTR1AADRA1DADRA1AADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2008526700-A 2008-07-24 JP claimed
EP-1761524-A1 PHENYL DIAZEPANE CARBOXAMIDES AND ANNELATED PHENYL PIPERAZINE CARBOXAMIDES CONTAINING OXYGEN AND USED AS DOPAMINE D3 ANTAGONISTS SCHWARZ PHARMA AG (DE) 2007-03-14 EP claimed
WO-2006072430-A1 PHENYL DIAZEPANE CARBOXAMIDES AND ANNELATED PHENYL PIPERAZINE CARBOXAMIDES CONTAINING OXYGEN AND USED AS DOPAMINE D3 ANTAGONISTS SCHWARZ PHARMA AG (DE) 2006-07-13 WO claimed