SCHEMBL5099611

SCHEMBL5099611

O=C(O)c1c(Br)cccc1-c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
MAPK1 P28482 1/20 0.56
FOLH1 Q04609 3/20 0.53
HNF4A P41235 1/20 0.48
AKR1C3 P42330 2/20 0.43
AKR1C2 P52895 2/20 0.43
AKR1C1 Q04828 2/20 0.43
PRNP P04156 1/20 0.43
KMT2A Q03164 2/20 0.43
FABP4 P15090 2/20 0.42
BCAT2 O15382 1/20 0.42
FABP3 P05413 1/20 0.41
FABP5 Q01469 1/20 0.41
AKR1C4 P17516 1/20 0.41
HTT P42858 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29501734 0.90 ALDH1A1 (0.59) ALDH1A1MAPK1FOLH1HNF4AAKR1C3
SCHEMBL11816433 0.88 ALDH1A1 (0.48) ALDH1A1MAPK1FOLH1HNF4AAKR1C3
SCHEMBL6536482 0.85 ALDH1A1 (0.43) ALDH1A1MAPK1FOLH1AKR1C3AKR1C2
SCHEMBL593127 0.85 FOLH1 (0.61) ALDH1A1FOLH1HNF4AKMT2AFABP4
SCHEMBL26554906 0.85 BCAT2 (0.53) ALDH1A1MAPK1FOLH1HNF4AAKR1C3
SCHEMBL15824265 0.85 ALDH1A1 (0.52) ALDH1A1MAPK1FOLH1HNF4AAKR1C3
SCHEMBL27542139 0.84 AKR1C3 (0.49) ALDH1A1MAPK1FOLH1HNF4AAKR1C3
SCHEMBL851906 0.80 HTT (0.53) ALDH1A1MAPK1KMT2AHTTCA12
SCHEMBL570378 0.80 CA12 (0.52) ALDH1A1AKR1C3AKR1C2AKR1C1PRNP
SCHEMBL28712874 0.79 ALDH1A1 (0.51) ALDH1A1MAPK1FOLH1HNF4AAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240389450-A1 LIGHT EMITTING ELEMENT, PRODUCTION METHOD FOR LIGHT EMITTING ELEMENT, DISPLAY DEVICE, AND PRODUCTION METHOD FOR DISPLAY DEVICE Sharp Display Technology Corporation (JP) 2024-11-21 US claimed
WO-2023079616-A1 LIGHT EMITTING ELEMENT, PRODUCTION METHOD FOR LIGHT EMITTING ELEMENT, DISPLAY DEVICE, AND PRODUCTION METHOD FOR DISPLAY DEVICE シャープディスプレイテクノロジー株式会社 2023-05-11 WO claimed
US-20240389450-A1 LIGHT EMITTING ELEMENT, PRODUCTION METHOD FOR LIGHT EMITTING ELEMENT, DISPLAY DEVICE, AND PRODUCTION METHOD FOR DISPLAY DEVICE Sharp Display Technology Corporation (JP) 2024-11-21 US disclosed
US-20230331675-A1 AROMATIC ETHYLENE COMPOUND AND PREPARATION METHOD THEREFOR, AND INTERMEDIATE, PHARMACEUTICAL COMPOSITION, AND APPLICATION THEREOF GUANGZHOU MAXINOVEL PHARMACEUTICALS CO., LTD. (CN) 2023-10-19 US disclosed
US-20230331675-A1 AROMATIC ETHYLENE COMPOUND AND PREPARATION METHOD THEREFOR, AND INTERMEDIATE, PHARMACEUTICAL COMPOSITION, AND APPLICATION THEREOF GUANGZHOU MAXINOVEL PHARMACEUTICALS CO., LTD. (CN) 2023-10-19 US disclosed
EP-4212511-A1 AROMATIC ETHYLENE COMPOUND AND PREPARATION METHOD THEREFOR, AND INTERMEDIATE, PHARMACEUTICAL COMPOSITION, AND APPLICATION THEREOF Guangzhou Maxinovel Pharmaceuticals Co., Ltd. (CN) 2023-07-19 EP disclosed
WO-2023079616-A1 LIGHT EMITTING ELEMENT, PRODUCTION METHOD FOR LIGHT EMITTING ELEMENT, DISPLAY DEVICE, AND PRODUCTION METHOD FOR DISPLAY DEVICE シャープディスプレイテクノロジー株式会社 2023-05-11 WO disclosed
CN-112552154-B Preparation method of 1-bromofluorenone 河南省科学院化学研究所有限公司 2022-09-09 CN disclosed
WO-2022052926-A1 AROMATIC ETHYLENE COMPOUND AND PREPARATION METHOD THEREFOR, AND INTERMEDIATE, PHARMACEUTICAL COMPOSITION, AND APPLICATION THEREOF 广州再极医药科技有限公司 2022-03-17 WO disclosed
CN-112552154-A Preparation method of 1-bromofluorenone 河南省科学院化学研究所有限公司 2021-03-26 CN disclosed
US-20150318498-A1 Metal Complexes MERCK PATENT GMBH (DE) 2015-11-05 US disclosed
CN-104870460-A Metal complexes MERCK PATENT GMBH 2015-08-26 CN disclosed
US-7446222-B2 Phenyl compounds GLAXO GROUP LIMITED (GB) 2008-11-04 US disclosed
US-20060235057-A1 Phenyl compounds GLAXO GROUP LIMITED (GB) 2006-10-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060235057-A1 Phenyl compounds RXRB, CYP2C9, RXFP1 ALDH1A1 1584/4885MAPK1 2875/4885FOLH1 3524/4885
US-20150318498-A1 Metal Complexes SOD1, AP1M1, AP3M1 ALDH1A1 3721/4885MAPK1 4229/4885FOLH1 4517/4885
US-20230331675-A1 AROMATIC ETHYLENE COMPOUND AND PREPARATION METHOD THEREFOR, AND INTERMEDIATE, PHARMACEUTICAL COMPOSITION, AND APPLICATION THEREOF PDCD1, CD274, PDCD1LG2 ALDH1A1 243/4885MAPK1 353/4885FOLH1 2750/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.