SCHEMBL5111766

SCHEMBL5111766

Cc1cc(C)c(N2CCCC2)c(C)c1NS(=O)(=O)c1cccc2cccnc12

nearest known ligand 0.63

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GFER P55789 1/20 0.59
MEN1 O00255 4/20 0.54
KMT2A Q03164 4/20 0.54
SLC40A1 Q9NP59 3/20 0.51
MAPT P10636 1/20 0.51
TSHR P16473 2/20 0.50
ALOX15 P16050 1/20 0.50
ATM Q13315 1/20 0.49
TP53 P04637 1/20 0.47
HTT P42858 1/20 0.47
ALDH1A1 P00352 2/20 0.46
GAA P10253 1/20 0.46
PKM P14618 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL533550 0.82 HCRTR1 (0.47) MEN1KMT2AMAPTTSHRTP53
SCHEMBL532980 0.81 JAK2 (0.48) GFERMEN1KMT2ASLC40A1MAPT
SCHEMBL532939 0.78 EDNRA (0.43) GFERMEN1KMT2AMAPTALDH1A1
SCHEMBL532038 0.78 ALDH1A1 (0.54) GFERKMT2ASLC40A1MAPTTSHR
SCHEMBL534052 0.78 MEN1 (0.47) MEN1KMT2AMAPTTSHRALDH1A1
SCHEMBL533512 0.77 SLC22A12 (0.44) MEN1KMT2ASLC40A1MAPTTSHR
SCHEMBL533083 0.76 EDNRA (0.46) MAPTALDH1A1
SCHEMBL6363732 0.75 GFER (0.98) GFERMEN1KMT2AMAPTTSHR
SCHEMBL532999 0.75 TP53 (0.48) MEN1KMT2ATP53ALDH1A1CYP3A4
SCHEMBL532998 0.75 JAK2 (0.37) GFERMEN1KMT2AMAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed