SCHEMBL5118839

SCHEMBL5118839

CCCCNc1c(N)cnc2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 1/20 0.49
LMNA P02545 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
ACP1 P24666 1/20 0.48
HRH3 Q9Y5N1 2/20 0.47
SLC2A1 P11166 6/20 0.47
TLR8 Q9NR97 1/20 0.47
CACNA2D1 P54289 1/20 0.45
POLB P06746 2/20 0.44
RAD52 P43351 2/20 0.44
KMT2A Q03164 2/20 0.44
NPC1 O15118 1/20 0.44
APOBEC3A P31941 1/20 0.44
RAB9A P51151 1/20 0.44
APOBEC3G Q9HC16 1/20 0.44
MEN1 O00255 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31197371 0.94 S1PR2 (0.57) S1PR2LMNASMN1; SMN2NPSR1CYP1A2
SCHEMBL10589295 0.94 S1PR2 (0.57) S1PR2LMNASMN1; SMN2NPSR1CYP1A2
SCHEMBL9602243 0.94 S1PR2 (0.57) S1PR2LMNASMN1; SMN2NPSR1CYP1A2
SCHEMBL18843434 0.91 APP (0.50) S1PR2LMNASMN1; SMN2NPSR1CYP1A2
SCHEMBL6096807 0.89 HTR1A (0.51) HRH3SLC2A1POLBRAD52
SCHEMBL7218710 0.87 POLB (0.45) LMNAHRH3SLC2A1CACNA2D1POLB
SCHEMBL6787115 0.85 HRH3 (0.45) HRH3SLC2A1CACNA2D1POLBRAD52
SCHEMBL10728537 0.85 POLB (0.63) LMNASMN1; SMN2HRH3SLC2A1POLB
SCHEMBL4336578 0.85 POLB (0.44) LMNAHRH3SLC2A1CACNA2D1POLB
SCHEMBL9837697 0.84 MEN1 (0.42) CYP1A2HRH3KMT2AMEN1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080015184-A1 Urea Substituted Imidazopyridines, Imidazoquinolines, and Imidazonaphthyridines 3M INNOVATIVE PROPERTIES COMPANY (US) 2008-01-17 US disclosed
EP-1701955-A1 ARYLALKENYL AND ARYLALKYNYL SUBSTITUTED IMIDAZOQUINOLINES 3M Innovative Properties Company (US) 2006-09-20 EP disclosed
WO-2005123079-A2 UREA SUBSTITUTED IMIDAZOPYRIDINES, IMIDAZOQUINOLINES, AND IMIDAZONAPHTHYRIDINES 3M INNOVATIVE PROPERTIES COMPANY (US) 2005-12-29 WO disclosed
WO-2005066170-A1 ARYLALKENYL AND ARYLALKYNYL SUBSTITUTED IMIDAZOQUINOLINES 3M INNOVATIVE PROPERTIES COMPANY (US) 2005-07-21 WO disclosed
US-4698348-A 1H-imidazo[4,5-c]quinolines and their use as bronchodilating agents RIKER LABORATORIES, INC. (US) 1987-10-06 US disclosed
US-4689338-A 1H-Imidazo[4,5-c]quinolin-4-amines and antiviral use RIKER LABORATORIES, INC. (US) 1987-08-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080015184-A1 Urea Substituted Imidazopyridines, Imidazoquinolines, and Imidazonaphthyridines IL2, EIF2AK2, IL4 S1PR2 3970/4885LMNA 3978/4885SMN1; SMN2 3238/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.