SCHEMBL5118879

SCHEMBL5118879

CC(C)(C)OC(=O)N1CCC(NC(=O)CCl)C1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.53
USP30 Q70CQ3 9/20 0.53
HSD11B1 P28845 6/20 0.50
CYP2C9 P11712 1/20 0.50
HDAC4 P56524 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
PARP1 P09874 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18632877 1.00 EPHX1 (0.53) EPHX1USP30HSD11B1CYP2C9HDAC4
SCHEMBL30505540 1.00 EPHX1 (0.53) EPHX1USP30HSD11B1CYP2C9HDAC4
SCHEMBL13636132 0.92 USP30 (0.55) EPHX1USP30HSD11B1CYP2C9HDAC4
SCHEMBL25948405 0.92 USP30 (0.55) EPHX1USP30HSD11B1CYP2C9HDAC4
SCHEMBL25948398 0.92 USP30 (0.55) EPHX1USP30HSD11B1CYP2C9HDAC4
SCHEMBL4206232 0.92 EPHX1 (0.63) EPHX1HDAC4PARP1
SCHEMBL25245907 0.88 NR1H2 (0.48) EPHX1USP30
SCHEMBL17560314 0.87 EPHX1 (0.55) EPHX1USP30HSD11B1CYP2C9HDAC4
SCHEMBL2040388 0.87 EPHX1 (0.55) EPHX1USP30HSD11B1CYP2C9HDAC4
SCHEMBL17560313 0.87 EPHX1 (0.55) EPHX1USP30HSD11B1CYP2C9HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080300232-A1 N-Piperidine Derivatives as Ccr3 Modulators ASTRAZENECA AB (SE) 2008-12-04 US disclosed
EP-1730136-A1 N-PIPERIDINE DERIVATES AS CCR3 MODULATORS AstraZeneca AB (SE) 2006-12-13 EP disclosed
WO-2005090330-A1 N-PIPERIDINE DERIVATES AS CCR3 MODULATORS ASTRAZENECA AB (SE) 2005-09-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080300232-A1 N-Piperidine Derivatives as Ccr3 Modulators CCR3, CCR1, CCR4 EPHX1 1340/4885USP30 1342/4885HSD11B1 2053/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.