SCHEMBL5126595

SCHEMBL5126595

CCc1cccc(CN(C[C@@H](O)[C@@H](N)Cc2cc(F)cc(F)c2)C(=O)CCC(=O)Nc2ccc(F)c(Cl)c2)c1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.41
TSHR P16473 2/20 0.40
KDM4E B2RXH2 2/20 0.39
MAPT P10636 3/20 0.39
BACE1 P56817 3/20 0.38
CTSD P07339 2/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5130327 0.89 BACE1 (0.40) LMNAMAPTBACE1CTSDSMN1; SMN2
SCHEMBL5120761 0.88 ALDH1A1 (0.40) LMNAMAPTBACE1CTSDMEN1
SCHEMBL5120921 0.87 HTT (0.42) TSHRMAPTBACE1CTSDMEN1
SCHEMBL5579835 0.83 PPARA (0.38) LMNABACE1CTSDMEN1KMT2A
SCHEMBL5125902 0.83 KMT2A (0.41) LMNAMAPTBACE1CTSDMEN1
SCHEMBL5125566 0.82 GRM5 (0.41) BACE1CTSDKMT2ASMN1; SMN2NPC1
SCHEMBL5127424 0.81 KMT2A (0.44) KDM4EBACE1CTSDMEN1KMT2A
SCHEMBL5120573 0.81 BACE1 (0.40) BACE1CTSD
SCHEMBL5130529 0.81 CTSD (0.39) TSHRBACE1CTSDMEN1KMT2A
SCHEMBL5118334 0.80 BACE1 (0.41) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080161325-A1 e.g. N1-[3-amino-4-(3,5-difluorophenyl)-2-hydroxybutyl]-3-(butylsulfonyl)-N1-(3-ethylbenzyl)-D-alaninamide dihydrochloride; inhibitors of amyloid beta-secretase enzyme; neurodegenerative diseases: Alzheimer's, Parkinson's diseases, Down's syndrome ELAN PHARMACEUTICALS, INC. 2008-07-03 US disclosed
US-7294642-B2 1,3-Diamino-2-hydroxypropane pro-drug derivatives ELAN PHARMACEUTICALS, INC. (US) 2007-11-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080161325-A1 e.g. N1-[3-amino-4-(3,5-difluorophenyl)-2-hydroxybutyl]-3-(butylsulfonyl)-N1-(3-ethylbenzyl)-D-alaninamide dihydrochloride; inhibitors of amyloid beta-secretase enzyme; neurodegenerative diseases: Alzheimer's, Parkinson's diseases, Down's syndrome BACE1, APP, BACE2 LMNA 133/4885TSHR 4721/4885KDM4E 3054/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.