SCHEMBL5128262

SCHEMBL5128262

COCCNCCc1cc[c]cc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.40
KDM4E B2RXH2 4/20 0.39
RECQL P46063 1/20 0.39
ADRB2 P07550 2/20 0.38
ALDH1A1 P00352 4/20 0.38
PKM P14618 1/20 0.37
SIGMAR1 Q99720 6/20 0.37
KCNH2 Q12809 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
HTT P42858 1/20 0.36
DRD2 P14416 1/20 0.35
DRD1 P21728 1/20 0.35
DRD4 P21917 1/20 0.35
DRD3 P35462 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5131567 0.89 KMT2A (0.43) GAAKDM4EALDH1A1SIGMAR1MEN1
SCHEMBL1033166 0.83 L3MBTL1 (0.57) L3MBTL1KDM4ERECQLADRB2ALDH1A1
SCHEMBL7235032 0.81 GAA (0.65) GAAKDM4EADRB2SIGMAR1KCNH2
SCHEMBL198568 0.80 NR3C1 (0.36) KDM4EADRB2
SCHEMBL28152391 0.80 GAA (0.42) GAAL3MBTL1KDM4ERECQLADRB2
SCHEMBL29602871 0.78 TAAR1 (0.55) GAAL3MBTL1KDM4ERECQLALDH1A1
SCHEMBL14566080 0.78 TAAR1 (0.55) L3MBTL1KDM4EALDH1A1KCNH2KMT2A
SCHEMBL28291658 0.76 SIGMAR1 (0.41) GAAL3MBTL1SIGMAR1
SCHEMBL7003569 0.76 IDO1 (0.38) L3MBTL1KDM4EALDH1A1PKMKCNH2
SCHEMBL7002413 0.75 L3MBTL1 (0.37) L3MBTL1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008020203-A1 PYRIDINYLQUINAZ0LINAMINE DERIVATIVES AND THEIR USE AS B-RAF INHIBITORS ASTRAZENECA AB (SE) 2008-02-21 WO disclosed