SCHEMBL5129596

SCHEMBL5129596

CONC(=O)c1ccc(-c2ccc3nc(N)nc(OCCF)c3c2)cc1.Nc1nc(OCCF)c2cc(-c3ccc(C(=O)N4CCSC4)cc3)ccc2n1.Nc1nc(OCCF)c2cc(-c3ccc(C(=O)N4CCSCC4)cc3)ccc2n1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.35
GABRA5 P31644 2/20 0.34
JAK1 P23458 1/20 0.34
LIPC P11150 3/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
S1PR1 P21453 1/20 0.33
S1PR3 Q99500 1/20 0.33
MAPKAPK2 P49137 1/20 0.33
CCNC P24863 1/20 0.32
CDK8 P49336 1/20 0.32
SCD O00767 1/20 0.32
DPP4 P27487 1/20 0.32
LIPG Q9Y5X9 1/20 0.32
MGLL Q99685 1/20 0.32
SYK P43405 1/20 0.32
GSK3B P49841 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5140172 0.98 GABRA5 (0.35) HPGDGABRA5JAK1LIPCALDH1A1
SCHEMBL5131336 0.94 GABRA5 (0.36) HPGDGABRA5JAK1LIPCALDH1A1
SCHEMBL3331181 0.91 DPP4 (0.37) HPGDGABRA5JAK1S1PR1S1PR3
SCHEMBL3338041 0.90 HPGD (0.40) HPGDGABRA5JAK1ALDH1A1HSD17B10
SCHEMBL3335512 0.86 DPP4 (0.38) HPGDGABRA5JAK1S1PR1S1PR3
SCHEMBL3335323 0.85 ALDH1A1 (0.40) ALDH1A1CYP3A4TSHRHSD17B10S1PR1
SCHEMBL3337282 0.83 MGLL (0.41) HPGDGABRA5JAK1ALDH1A1HSD17B10
SCHEMBL3336025 0.81 HPGD (0.45) HPGD
SCHEMBL3333969 0.81 HPGD (0.43) HPGDJAK1ALDH1A1HSD17B10MGLL
SCHEMBL3341492 0.80 ALDH1A1 (0.39) ALDH1A1CYP3A4TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009077-A2 4,6-DL- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO disclosed