SCHEMBL5132852

SCHEMBL5132852

CS(=O)(=O)c1nc2cc(C#N)c(Cl)nc2n1S(C)(=O)=O

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
KHK P50053 1/20 0.34
NPSR1 Q6W5P4 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
HPGD P15428 1/20 0.33
PGK1 P00558 1/20 0.31
GLA P06280 1/20 0.30
POLB P06746 1/20 0.30
GAA P10253 1/20 0.30
XBP1 P17861 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5043253 0.68 ALDH1A1 (0.43) ALDH1A1KHKNPSR1CYP1A2CYP2C9
SCHEMBL10803255 0.65 ALDH1A1 (0.42) ALDH1A1KHKNPSR1CYP1A2CYP2C9
SCHEMBL566209 0.62 KHK (0.57) ALDH1A1KHKNPSR1CYP1A2CYP2C9
SCHEMBL10832908 0.61 SMN1; SMN2 (0.33) SMN1; SMN2KDM4EGAA
SCHEMBL23357368 0.61 ALDH1A1 (0.41) ALDH1A1KHKNPSR1CYP1A2CYP2C9
SCHEMBL30711996 0.61 ALDH1A1 (0.41) ALDH1A1KHKNPSR1CYP1A2CYP2C9
SCHEMBL3554942 0.61 CSNK1A1 (0.40) ALDH1A1KHKNPSR1CYP1A2CYP2C9
SCHEMBL33527400 0.60 ALDH1A1 (0.41) ALDH1A1KHKNPSR1CYP1A2CYP2C9
SCHEMBL33527205 0.59 LMNA (0.53) ALDH1A1KHKNPSR1CYP1A2CYP2C9
SCHEMBL6493251 0.59 ALDH1A1 (0.50) ALDH1A1KHKNPSR1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981342-A1 SELECTIVE BENZYLAMINE DERIVATIVES AND THEIR UTILITY AS CHOLESTEROL ESTER-TRANSFER PROTEIN INHIBITORS Reddy US Therapeutics, Inc. (US) 2008-10-22 EP disclosed
WO-2007075194-A1 SELECTIVE BENZYLAMINE DERIVATIVES AND THEIR UTILITY AS CHOLESTEROL ESTER-TRANSFER PROTEIN INHIBITORS REDDY US THERAPEUTICS, INC. (US) 2007-07-05 WO disclosed