SCHEMBL5133315

SCHEMBL5133315

O=C(c1ccc2[nH]c(-c3ccc(Cl)c4c[nH]cc34)cc2c1)N1CCCC(O)C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.46
MRGPRX4 Q96LA9 1/20 0.39
JAK2 O60674 1/20 0.38
CCNC P24863 1/20 0.38
CDK8 P49336 1/20 0.38
SLC40A1 Q9NP59 1/20 0.38
GRM3 Q14832 1/20 0.38
HPGD P15428 1/20 0.37
ROCK2 O75116 2/20 0.37
KMT2A Q03164 1/20 0.36
DYRK3 O43781 1/20 0.36
RPS6KB1 P23443 1/20 0.36
CLK2 P49760 1/20 0.36
ROCK1 Q13464 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
CSNK1G1 Q9HCP0 1/20 0.36
STK17A Q9UEE5 1/20 0.36
MAPT P10636 1/20 0.36
PDK2 Q15119 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5133467 0.89 KDR (0.47) KDRSLC40A1HPGDMGLL
SCHEMBL3033406 0.81 KDR (0.45) KDRMRGPRX4JAK2SLC40A1GRM3
SCHEMBL5133013 0.73 CHEK1 (0.47)
SCHEMBL5076120 0.71 KDR (0.80) KDRPDK2MGLL
SCHEMBL3049984 0.71 KDR (0.43) KDRGRM3PDK2
SCHEMBL3047646 0.70 KDR (0.45) KDRSLC40A1MGLL
SCHEMBL5050597 0.69 HTT (0.45) HPGD
SCHEMBL5133622 0.69 TERT (0.44) HPGDKMT2AMAPT
SCHEMBL5134254 0.69 NPC1 (0.41) KDRHPGDKMT2AMAPT
SCHEMBL3047573 0.68 KDR (0.46) KDRHPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed