SCHEMBL5133467

SCHEMBL5133467

O=C(c1ccc2[nH]c(-c3ccc(Cl)c4c[nH]cc34)cc2c1)N1CCC(O)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.47
SLC40A1 Q9NP59 1/20 0.41
CCR3 P51677 1/20 0.41
EIF4E P06730 1/20 0.40
MGLL Q99685 2/20 0.40
CYP51A1 Q16850 2/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
OXTR P30559 1/20 0.38
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
HTR1A P08908 1/20 0.38
HPGD P15428 1/20 0.38
HRH4 Q9H3N8 1/20 0.38
HSD11B1 P28845 1/20 0.38
LRRK2 Q5S007 1/20 0.37
MAPK14 Q16539 1/20 0.37
CCNA2 P20248 1/20 0.37
CDK2 P24941 1/20 0.37
TTK P33981 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5133315 0.89 KDR (0.46) KDRSLC40A1MGLLHPGD
SCHEMBL3047646 0.80 KDR (0.45) KDRSLC40A1CCR3EIF4EMGLL
SCHEMBL5133013 0.80 CHEK1 (0.47)
SCHEMBL5753668 0.73 KDR (0.45) KDRMGLLHSP90AA1HSP90AB1OXTR
SCHEMBL5133476 0.72 HPGD (0.50) HPGD
SCHEMBL5133622 0.71 TERT (0.44) HPGD
SCHEMBL5134254 0.71 NPC1 (0.41) KDRHPGDHRH4
Hydrochloric Acid SCHEMBL3047329 0.71 KDR (0.52) KDRCCR3MGLLOXTR
SCHEMBL3047974 0.71 KDR (0.44) KDRCCR3HTR1A
SCHEMBL5133818 0.70 MAOA (0.47) HSP90AA1HSP90AB1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed