SCHEMBL5133804

SCHEMBL5133804

CC(C)(C)OC(=O)NCCCOc1ccc(-c2cc3cc(CN4CCN(CCO)CC4)ccc3n2C(=O)OC(C)(C)C)c2c[nH]cc12

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.36
NR1H2 P55055 3/20 0.36
SUCNR1 Q9BXA5 1/20 0.36
SIGMAR1 Q99720 2/20 0.35
MAPK1 P28482 1/20 0.35
BRD4 O60885 1/20 0.35
ATR Q13535 2/20 0.34
ATRIP Q8WXE1 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27700342 0.87 DRD2 (0.33) DRD2NR1H2SUCNR1SIGMAR1MAPK1
SCHEMBL3037100 0.87 DRD2 (0.34) DRD2NR1H2SUCNR1SIGMAR1MAPK1
SCHEMBL3037188 0.79 PARP1 (0.36) NR1H2
SCHEMBL5048352 0.76 PARP1 (0.34) NR1H2ATR
SCHEMBL5140104 0.76 NR1H2 (0.34) NR1H2ATRATRIP
SCHEMBL3052537 0.74 PARP1 (0.35) NR1H2
SCHEMBL3046855 0.74 NR1H2 (0.39) NR1H2BRD4ATRATRIP
SCHEMBL3043944 0.74 PARP1 (0.35) NR1H2ATR
SCHEMBL3144005 0.74 NR1H2 (0.38) NR1H2SUCNR1BRD4ATRATRIP
SCHEMBL27700218 0.73 NR1H2 (0.33) NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed