SCHEMBL5134530

SCHEMBL5134530

Cc1c(F)c(C(N)=O)c(CC2CCOCC2)c(C2CCNCC2)c1F

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.33
EED O75530 1/20 0.31
RBBP4 Q09028 1/20 0.31
SUZ12 Q15022 1/20 0.31
EZH2 Q15910 1/20 0.31
AEBP2 Q6ZN18 1/20 0.31
BTK Q06187 2/20 0.31
OPRL1 P41146 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5146834 0.72 KMT2A (0.32)
SCHEMBL5190879 0.72 IRAK4 (0.36) PARP1BTK
SCHEMBL5134855 0.66 OPRL1 (0.34) BTKOPRL1
SCHEMBL5136172 0.66 IRAK4 (0.38) PARP1
SCHEMBL5134806 0.65 PARP2 (0.39) PARP1BTK
SCHEMBL5135452 0.59 SLC6A4 (0.47) PARP1EZH2
SCHEMBL14168394 0.58 POLB (0.44)
SCHEMBL11044013 0.58 TAS1R3 (0.45)
SCHEMBL17185049 0.58 PARP1 (0.46) PARP1
SCHEMBL2311682 0.57 TAS1R3 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942893-A2 PIPERIDINE GLYCINE TRANSPORTER INHIBITORS Merck & Co., Inc. (US) 2008-07-16 EP disclosed
WO-2007053400-A2 PIPERIDINE GLYCINE TRANSPORTER INHIBITORS MERCK & CO., INC. (US) 2007-05-10 WO disclosed