SCHEMBL5146834

SCHEMBL5146834

Cc1c(F)c(C(N)=O)c(CC2CCCO2)c(C2CCNCC2)c1C(F)(F)F

nearest known ligand 0.32

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.32
KDM4E B2RXH2 3/20 0.31
ALDH1A1 P00352 3/20 0.31
GAA P10253 2/20 0.31
MAPK1 P28482 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
HPGD P15428 2/20 0.30
GLA P06280 1/20 0.30
PSEN1 P49768 2/20 0.30
PSEN2 P49810 2/20 0.30
APH1B Q8WW43 2/20 0.30
NCSTN Q92542 2/20 0.30
APH1A Q96BI3 2/20 0.30
PSENEN Q9NZ42 2/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5134124 0.83 KMT2A (0.34) KMT2AKDM4EALDH1A1HPGDMAPT
SCHEMBL5134530 0.72 PARP1 (0.33)
SCHEMBL5146827 0.65 CNR2 (0.41) HPGD
SCHEMBL5146830 0.64 ALDH1A1 (0.40) KMT2AKDM4EALDH1A1GAAMAPK1
SCHEMBL5134331 0.62 RAB9A (0.39) KMT2AKDM4EALDH1A1MAPK1NPSR1
SCHEMBL5134806 0.60 PARP2 (0.39)
SCHEMBL5134123 0.58 KMT2A (0.41) KMT2AKDM4EALDH1A1GAAMAPK1
SCHEMBL4763827 0.58 PARP1 (0.54) KMT2AKDM4EALDH1A1GAAHPGD
SCHEMBL5808501 0.56 HTR2C (0.44) KMT2A
SCHEMBL17594488 0.56 GABRA1 (0.34) KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942893-A2 PIPERIDINE GLYCINE TRANSPORTER INHIBITORS Merck & Co., Inc. (US) 2008-07-16 EP disclosed
WO-2007053400-A2 PIPERIDINE GLYCINE TRANSPORTER INHIBITORS MERCK & CO., INC. (US) 2007-05-10 WO disclosed