SCHEMBL5135172

SCHEMBL5135172

Cc1c(C(N)=O)cccc1C1(CC2CCOCC2)CCNCC1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 5/20 0.37
PARP1 P09874 9/20 0.36
PARP2 Q9UGN5 4/20 0.36
AURKA O14965 1/20 0.34
RPS6KB1 P23443 1/20 0.34
CNR1 P21554 3/20 0.33
CNR2 P34972 3/20 0.33
OPRL1 P41146 1/20 0.33
CCNC P24863 1/20 0.32
CDK8 P49336 1/20 0.32
HASPIN Q8TF76 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5135169 0.86 PARP1 (0.39) OPRM1PARP1PARP2AURKARPS6KB1
SCHEMBL5134855 0.76 OPRL1 (0.34) OPRL1
SCHEMBL5332677 0.74 OPRL1 (0.33) OPRL1
SCHEMBL30849224 0.68 PARP1 (0.40) OPRM1PARP1AURKA
SCHEMBL20822490 0.67 PARP1 (0.43) PARP1OPRL1
SCHEMBL25436221 0.66 PARP1 (0.41) PARP1PARP2AURKA
SCHEMBL5136172 0.65 IRAK4 (0.38) PARP1PARP2AURKARPS6KB1CNR1
SCHEMBL30343973 0.65 CCR2 (0.38) PARP1
SCHEMBL17185049 0.65 PARP1 (0.46) PARP1PARP2AURKARPS6KB1
SCHEMBL5190879 0.65 IRAK4 (0.36) PARP1CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942893-A2 PIPERIDINE GLYCINE TRANSPORTER INHIBITORS Merck & Co., Inc. (US) 2008-07-16 EP disclosed
WO-2007053400-A2 PIPERIDINE GLYCINE TRANSPORTER INHIBITORS MERCK & CO., INC. (US) 2007-05-10 WO disclosed