SCHEMBL5135181

SCHEMBL5135181

Nc1ccc(-n2ccc(NC(=O)c3ccc(N4CCN(C(=O)O)CC4)nc3)n2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.46
HDAC1 Q13547 6/20 0.44
ALDH1A1 P00352 2/20 0.43
MAPT P10636 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HDAC2 Q92769 3/20 0.42
HDAC3 O15379 3/20 0.42
DYRK1A Q13627 3/20 0.42
KCNH2 Q12809 3/20 0.40
RAB9A P51151 2/20 0.40
NPC1 O15118 1/20 0.40
KMT2A Q03164 1/20 0.40
HDAC10 Q969S8 2/20 0.39
WNT1 P04628 1/20 0.38
CLK2 P49760 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5135178 0.77 HDAC1 (0.51) HDAC1HDAC2HDAC3KCNH2RAB9A
SCHEMBL2456399 0.73 ME2 (0.47) LMNAALDH1A1MAPTSMN1; SMN2KDM4E
SCHEMBL4536729 0.71 HRH3 (0.55) ALDH1A1RAB9ANPC1KMT2A
SCHEMBL5134342 0.70 KMT2A (0.44) LMNAHDAC1ALDH1A1MAPTSMN1; SMN2
SCHEMBL5134339 0.70 KMT2A (0.44) LMNAHDAC1ALDH1A1MAPTSMN1; SMN2
SCHEMBL5183437 0.69 NPC1 (0.62) LMNAALDH1A1MAPTSMN1; SMN2KDM4E
SCHEMBL20339428 0.68 KMT2A (0.74) ALDH1A1MAPTKDM4ERAB9ANPC1
SCHEMBL14651869 0.67 RAB9A (0.63) LMNAHDAC1ALDH1A1MAPTSMN1; SMN2
SCHEMBL6824130 0.66 ALDH1A1 (0.69) LMNAALDH1A1KDM4EHPGDHTT
SCHEMBL4069836 0.66 HDAC1 (0.72) HDAC1HDAC2HDAC3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945617-A2 HISTONE DEACETYLASE INHIBITORS WITH ARYL-PYRAZOLYL MOTIFS Merck & Co., Inc. (US) 2008-07-23 EP disclosed
WO-2007055941-A2 HISTONE DEACETYLASE INHIBITORS WITH ARYL-PYRAZOLYL MOTIFS MERCK & CO., INC. (US) 2007-05-18 WO disclosed