SCHEMBL5135370

SCHEMBL5135370

COc1ccc(N(C)C2=CC(=O)C(N)=C(c3ncnc4ccccc34)C2=O)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.47
CSF1R P07333 2/20 0.41
HDAC1 Q13547 4/20 0.40
HDAC8 Q9BY41 4/20 0.40
HDAC6 Q9UBN7 4/20 0.40
CASP1 P29466 1/20 0.40
CASP14 P31944 1/20 0.40
CASP3 P42574 1/20 0.40
CASP2 P42575 1/20 0.40
CASP4 P49662 1/20 0.40
CASP5 P51878 1/20 0.40
CASP7 P55210 1/20 0.40
CASP9 P55211 1/20 0.40
CASP6 P55212 1/20 0.40
CASP8 Q14790 1/20 0.40
CASP12 Q6UXS9 1/20 0.40
CASP10 Q92851 1/20 0.40
EGFR P00533 4/20 0.39
KDR P35968 3/20 0.39
PDGFRB P09619 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5135369 0.93 CES1 (0.48) CES1CSF1RHDAC1HDAC8HDAC6
SCHEMBL5135024 0.74 ADORA2A (0.43) EGFRNPC1RAB9ASMN1; SMN2ADORA2A
SCHEMBL5135030 0.72 GAPDH (0.42) CES1EGFRKDRPDGFRBNPC1
SCHEMBL5664809 0.72 LDHA (0.40) KDRNPC1RAB9AADORA2A
SCHEMBL3112121 0.70 EGFR (0.72) CSF1RHDAC1HDAC8HDAC6CASP1
SCHEMBL5135022 0.68 ADORA2A (0.44) EGFRNPC1RAB9ASMN1; SMN2ADORA2A
SCHEMBL28872954 0.67 ADORA2A (0.66) EGFRKDRNPC1HTTRAB9A
SCHEMBL18774826 0.67 HTT (0.52) EGFRKDRNPC1HTTRAB9A
SCHEMBL5664944 0.65 KDR (0.43) EGFRKDR
SCHEMBL5134739 0.63 MAP4K4 (0.40) NPC1HTTRAB9ASMN1; SMN2ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080268460-A1 Assays to Identify Irreversibly Binding Inhibitors of Receptor Tyrosine Kinases WYETH (US) 2008-10-30 US disclosed