SCHEMBL5138879

SCHEMBL5138879

COc1cccc(-c2cccc(C3(C)Cc4ccccc4C(NOC(=O)C(F)(F)F)=N3)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 15/20 0.46
KCNH2 Q12809 6/20 0.43
LMNA P02545 3/20 0.38
HDAC6 Q9UBN7 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5030127 0.92 BACE1 (0.36) BACE1KCNH2LMNACYP1A2CYP3A4
SCHEMBL5025791 0.89 BACE1 (0.47) BACE1KCNH2LMNAHDAC6CYP1A2
SCHEMBL5028464 0.88 LMNA (0.40) BACE1KCNH2LMNAHDAC6CYP1A2
SCHEMBL5028541 0.82 BACE1 (0.56) BACE1LMNAHDAC6CYP1A2CYP3A4
Trifluoroacetic Acid SCHEMBL5001506 0.81 BACE1 (0.52) BACE1KCNH2LMNA
SCHEMBL2085929 0.78 BACE1 (0.42) BACE1KCNH2LMNAHDAC6HTT
SCHEMBL2085924 0.77 BACE1 (0.47) BACE1KCNH2HDAC6
SCHEMBL8240666 0.76 BACE1 (0.58) BACE1KCNH2
SCHEMBL5025594 0.75 LMNA (0.40) BACE1LMNAHDAC6
SCHEMBL2084752 0.75 BACE1 (0.40) BACE1KCNH2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957462-A2 NOVEL 2-AMINO-HETEROCYCLES UDEFUL IN THE TREATMENT OF ABETA-RELATED PATHOLOGIES Astra Zeneca AB (SE) 2008-08-20 EP disclosed
WO-2007058583-A2 NOVEL 2-AMINO-HETEROCYCLES USEFUL IN THE TREATMENT OF ABETA-RELATED PATHOLOGIES ASTRAZENECA AB (SE) 2007-05-24 WO disclosed