SCHEMBL5028541

SCHEMBL5028541

COc1cccc(-c2cccc(CCC3(C)Cc4ccccc4C(NOC(=O)C(F)(F)F)=N3)c2)c1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 10/20 0.56
LMNA P02545 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
NAMPT P43490 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5026434 0.85 BACE1 (0.41) BACE1CYP1A2CYP3A4CYP2C9CYP2C19
Trifluoroacetic Acid SCHEMBL5001971 0.84 BACE1 (0.68) BACE1LMNA
SCHEMBL5138879 0.82 BACE1 (0.46) BACE1LMNAHDAC6CYP1A2CYP3A4
SCHEMBL5025791 0.81 BACE1 (0.47) BACE1LMNAHDAC6CYP1A2CYP3A4
SCHEMBL5028464 0.80 LMNA (0.40) BACE1LMNAALDH1A1HDAC6CYP1A2
SCHEMBL8241111 0.79 BACE1 (0.62) BACE1
Trifluoroacetic Acid SCHEMBL5005126 0.74 BACE1 (0.57) BACE1LMNA
SCHEMBL5030127 0.74 BACE1 (0.36) BACE1LMNACYP1A2CYP3A4CYP2C9
SCHEMBL5025594 0.73 LMNA (0.40) BACE1LMNAALDH1A1HDAC6
SCHEMBL4997237 0.71 BACE1 (0.51) BACE1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957462-A2 NOVEL 2-AMINO-HETEROCYCLES UDEFUL IN THE TREATMENT OF ABETA-RELATED PATHOLOGIES Astra Zeneca AB (SE) 2008-08-20 EP claimed
WO-2007058583-A2 NOVEL 2-AMINO-HETEROCYCLES USEFUL IN THE TREATMENT OF ABETA-RELATED PATHOLOGIES ASTRAZENECA AB (SE) 2007-05-24 WO claimed