SCHEMBL5028464

SCHEMBL5028464

COc1cccc(-c2cccc(C3(C(F)(F)F)Cc4ccccc4C(NOC(=O)C(F)(F)F)=N3)c2)c1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.40
BACE1 P56817 12/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 1/20 0.38
KCNH2 Q12809 3/20 0.38
HDAC6 Q9UBN7 1/20 0.37
ALDH1A1 P00352 2/20 0.36
MAPK1 P28482 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5138879 0.88 BACE1 (0.46) LMNABACE1CYP1A2CYP3A4CYP2C9
SCHEMBL5025791 0.88 BACE1 (0.47) LMNABACE1CYP1A2CYP3A4CYP2C9
SCHEMBL5026581 0.83 MAPT (0.34) BACE1CYP1A2CYP3A4CYP2C9CYP2C19
Trifluoroacetic Acid SCHEMBL5001600 0.82 BACE1 (0.46) LMNABACE1KCNH2
SCHEMBL5028541 0.80 BACE1 (0.56) LMNABACE1CYP1A2CYP3A4CYP2C9
SCHEMBL8234584 0.80 BACE1 (0.47) BACE1KCNH2
SCHEMBL5030127 0.79 BACE1 (0.36) LMNABACE1CYP1A2CYP3A4CYP2C9
SCHEMBL2085929 0.78 BACE1 (0.42) LMNABACE1HTTKCNH2HDAC6
SCHEMBL2085924 0.76 BACE1 (0.47) BACE1KCNH2HDAC6
SCHEMBL5025594 0.75 LMNA (0.40) LMNABACE1HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957462-A2 NOVEL 2-AMINO-HETEROCYCLES UDEFUL IN THE TREATMENT OF ABETA-RELATED PATHOLOGIES Astra Zeneca AB (SE) 2008-08-20 EP disclosed
WO-2007058583-A2 NOVEL 2-AMINO-HETEROCYCLES USEFUL IN THE TREATMENT OF ABETA-RELATED PATHOLOGIES ASTRAZENECA AB (SE) 2007-05-24 WO disclosed