SCHEMBL5140093

SCHEMBL5140093

Clc1ccc(-c2cc(Cl)cc3c2OC(CNc2ccccc2)C3)c(Cl)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 3/20 0.58
EZH2 Q15910 1/20 0.46
NFKB1 P19838 2/20 0.43
NFKB2 Q00653 2/20 0.43
RELA Q04206 2/20 0.43
NPC1 O15118 4/20 0.34
RAB9A P51151 4/20 0.34
SMN1; SMN2 Q16637 4/20 0.34
ALDH1A1 P00352 2/20 0.34
HPGD P15428 2/20 0.34
TP53 P04637 1/20 0.34
TSHR P16473 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HSD17B10 Q99714 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
MAPK14 Q16539 1/20 0.34
CNR1 P21554 1/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4219176 0.83 AQP1 (0.80) AQP1EZH2NPC1RAB9ASMN1; SMN2
SCHEMBL5148358 0.82 NFKB1 (0.43) AQP1EZH2NFKB1NFKB2RELA
SCHEMBL4230701 0.82 AQP1 (0.58) AQP1EZH2NPC1RAB9ASMN1; SMN2
SCHEMBL4596987 0.81 SIRT2 (0.55) AQP1EZH2NPC1RAB9ASMN1; SMN2
SCHEMBL4220292 0.79 AQP1 (0.79) AQP1EZH2SIRT2HTR2AHTR2C
SCHEMBL4219183 0.77 AQP1 (0.65) AQP1EZH2SIRT2HTR2AHTR2C
SCHEMBL5140813 0.77 AQP1 (0.43) AQP1EZH2NFKB1NFKB2RELA
SCHEMBL4968974 0.76 AQP1 (0.54) AQP1EZH2NFKB1NFKB2RELA
SCHEMBL4225947 0.75 AQP1 (0.67) AQP1EZH2ALDH1A1NPSR1SIRT2
SCHEMBL6368238 0.75 AQP1 (0.47) AQP1EZH2NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871354-A1 TREATMENT OF PAIN Wyeth (US) 2008-01-02 EP disclosed
WO-2006116171-A1 TREATMENT OF PAIN WYETH (US) 2006-11-02 WO disclosed