SCHEMBL5148358

SCHEMBL5148358

Clc1ccc(Cl)c(-c2cccc3c2OC(CNc2ccccc2)C3)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 2/20 0.43
NFKB2 Q00653 2/20 0.43
RELA Q04206 2/20 0.43
AQP1 P29972 3/20 0.43
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
EZH2 Q15910 1/20 0.36
PRKAB2 O43741 2/20 0.35
PRKAG1 P54619 2/20 0.35
PRKAA2 P54646 2/20 0.35
PRKAA1 Q13131 2/20 0.35
PRKAG3 Q9UGI9 2/20 0.35
PRKAG2 Q9UGJ0 2/20 0.35
PRKAB1 Q9Y478 2/20 0.35
CHRM1 P11229 2/20 0.35
SENP1 Q9P0U3 1/20 0.35
CRHR1 P34998 1/20 0.34
MAPK14 Q16539 1/20 0.34
CHRM3 P20309 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596919 0.85 AQP1 (0.58) AQP1EZH2PRKAB2PRKAG1PRKAA2
SCHEMBL4230182 0.83 AQP1 (0.42) AQP1EZH2PRKAB2PRKAG1PRKAA2
SCHEMBL5140093 0.82 AQP1 (0.58) NFKB1NFKB2RELAAQP1NPC1
SCHEMBL4226043 0.81 AQP1 (0.56) AQP1EZH2PRKAB2PRKAG1PRKAA2
SCHEMBL5795152 0.81 AQP1 (0.56) AQP1EZH2PRKAB2PRKAG1PRKAA2
SCHEMBL4596728 0.81 SIRT2 (0.52) AQP1PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4964691 0.80 AQP1 (0.43) AQP1EZH2PRKAB2PRKAG1PRKAA2
SCHEMBL4964699 0.80 AQP1 (0.43) AQP1EZH2PRKAB2PRKAG1PRKAA2
SCHEMBL4968974 0.76 AQP1 (0.54) NFKB1NFKB2RELAAQP1NPC1
SCHEMBL4968887 0.76 AQP1 (0.41) AQP1EZH2PRKAB2PRKAG1PRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871354-A1 TREATMENT OF PAIN Wyeth (US) 2008-01-02 EP claimed
WO-2006116171-A1 TREATMENT OF PAIN WYETH (US) 2006-11-02 WO claimed