SCHEMBL5140381

SCHEMBL5140381

CCCCC(N)N1CCSC1

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DPP7 Q9UHL4 7/20 0.37
DPP4 P27487 6/20 0.37
DPP8 Q6V1X1 3/20 0.37
DPP9 Q86TI2 3/20 0.37
OPRM1 P35372 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7557605 0.82
SCHEMBL1615523 0.78 OPRM1 (0.39) DPP7DPP4DPP8DPP9OPRM1
SCHEMBL1615233 0.76 OPRM1 (0.48) OPRM1
SCHEMBL28298745 0.74 OPRM1 (0.46) OPRM1
SCHEMBL28298671 0.74 OPRM1 (0.46) OPRM1
SCHEMBL1615271 0.74 OPRM1 (0.46) OPRM1
SCHEMBL28300172 0.74 OPRM1 (0.46) OPRM1
SCHEMBL1614359 0.74 OPRM1 (0.46) OPRM1
SCHEMBL2914564 0.74 HRH3 (0.40) DPP7DPP4DPP8DPP9OPRM1
SCHEMBL1614413 0.74 OPRM1 (0.46) OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2055302-B1 Method for the improvement of islet signaling in diabetes mellitus and for its prevention ROYALTY PHARMA COLLECTION TRUST (US) 2014-09-10 EP claimed
EP-1283735-B2 METHOD FOR THE IMPROVEMENT OF ISLET SIGNALING IN DIABETES MELLITUS AND FOR ITS PREVENTION ROYALTY PHARMA COLLECTION TRUST (US) 2012-10-24 EP claimed
EP-1283735-B1 METHOD FOR THE IMPROVEMENT OF ISLET SIGNALING IN DIABETES MELLITUS AND FOR ITS PREVENTION PROSIDION LTD (GB) 2008-12-31 EP claimed