SCHEMBL5140700

SCHEMBL5140700

COc1cc(OC2CCN(C)C2)ccc1-c1cccc(Nc2ccccc2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 3/20 0.47
CDK2 P24941 1/20 0.47
CDK9 P50750 1/20 0.47
CDK5 Q00535 1/20 0.47
NOS3 P29474 1/20 0.46
NOS1 P29475 1/20 0.46
NOS2 P35228 1/20 0.46
TTK P33981 2/20 0.44
IGF1R P08069 3/20 0.43
INSR P06213 3/20 0.43
ALK Q9UM73 2/20 0.43
DYRK1B Q9Y463 1/20 0.41
GALR2 O43603 1/20 0.40
GALR1 P47211 1/20 0.40
AXL P30530 2/20 0.40
KDR P35968 1/20 0.40
PDE3B Q13370 2/20 0.40
PDE3A Q14432 2/20 0.40
PDE10A Q9Y233 2/20 0.40
MAP4K1 Q92918 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5145370 0.86 CDK2 (0.45) CDK2CDK9CDK5TTKIGF1R
SCHEMBL5134247 0.84 CDK2 (0.52) CHEK1CDK2CDK9CDK5IGF1R
SCHEMBL221344 0.82 NOS1 (0.65) CHEK1NOS3NOS1NOS2TTK
SCHEMBL5140699 0.81 NOS3 (0.53) CHEK1NOS3NOS1NOS2TTK
SCHEMBL16241884 0.78 CHEK1 (0.48) CHEK1CDK2NOS3NOS1NOS2
SCHEMBL221859 0.77 NOS1 (0.57) CHEK1CDK2NOS3NOS1NOS2
SCHEMBL27981858 0.76 CHEK1 (0.45) CHEK1NOS3NOS1NOS2IGF1R
SCHEMBL3546662 0.75 INSR (0.47) CHEK1TTKIGF1RINSRALK
SCHEMBL422148 0.74 NOS3 (0.47) CHEK1NOS3NOS1NOS2PDE3B
SCHEMBL424370 0.74 NOS1 (0.54) CHEK1NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1877054-A2 NICOTINAMIDE RIBOSIDE AND ANALOGUES THEREOF Sirtris Pharmaceuticals, Inc. (US) 2008-01-16 EP disclosed
WO-2006105440-A2 NICOTINAMIDE RIBOSIDE AND ANALOGUES THEREOF SIRTRIS PHARMACEUTICALS, INC. (US) 2006-10-05 WO disclosed