SCHEMBL5144590

SCHEMBL5144590

CC12CC3CC(C)(C1)CC(CC(=O)Nc1ncnc4c1CCN(Cc1ccc(F)cc1F)C4)(C3)C2

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GPR6 P46095 11/20 0.35
NTRK1 P04629 1/20 0.34
GRM2 Q14416 3/20 0.34
CYP2D6 P10635 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
ENPP2 Q13822 2/20 0.34
KCNK3 O14649 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4985493 0.91 EPHX2 (0.35) NTRK1GRM2
SCHEMBL4989382 0.90 LMNA (0.38) ALDH1A1
SCHEMBL4988694 0.89 EPHX2 (0.39) GPR6GRM2
SCHEMBL4982656 0.85 P2RX7 (0.38) ALDH1A1
SCHEMBL14272268 0.85 P2RX7 (0.40)
SCHEMBL5141408 0.85 P2RX7 (0.38)
SCHEMBL4991840 0.84 BRS3 (0.37) ALDH1A1
SCHEMBL5145755 0.83 P2RX7 (0.38) ALDH1A1
SCHEMBL14272270 0.82 EPHX2 (0.39)
SCHEMBL4985453 0.82 CXCR3 (0.47) GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7297700-B2 Bicycloheteroaryl compounds as P2X7 modulators and uses thereof RENOVIS, INC. (US) 2007-11-20 US claimed