SCHEMBL5144836

SCHEMBL5144836

O=c1ccnc(-c2cccs2)[nH]1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.55
PDE3A Q14432 1/20 0.55
GAA P10253 2/20 0.47
GFER P55789 1/20 0.47
KDM4E B2RXH2 5/20 0.46
HPGD P15428 4/20 0.46
PKM P14618 1/20 0.46
ALDH1A1 P00352 4/20 0.44
MEN1 O00255 2/20 0.44
MAPT P10636 2/20 0.44
KMT2A Q03164 2/20 0.44
LMNA P02545 1/20 0.44
GLA P06280 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
ERCC1 P07992 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1129657 0.72 ALDH1A1 (0.39) PDE3BPDE3AHPGDPKMALDH1A1
SCHEMBL11655 0.72 NISCH (0.48) GAAGFERKDM4EHPGDPKM
SCHEMBL10810557 0.71 PDE3B (1.00) PDE3BPDE3ACDK5CDK5R1TDO2
SCHEMBL1133436 0.69 GAA (0.50) PDE3BPDE3AGAAHPGDALDH1A1
SCHEMBL7454459 0.69 PDE3B (0.50) PDE3BPDE3AGAAHPGDALDH1A1
SCHEMBL17269663 0.69 GAA (0.47) GAAGFERKDM4EHPGDPKM
SCHEMBL18225434 0.68 GAA (0.54) GAAKDM4EHPGDALDH1A1MEN1
SCHEMBL28606824 0.68 NOTUM (0.48) PDE3BPDE3AGAAGFERKDM4E
SCHEMBL25754931 0.68 PIN1 (0.58) KDM4EHPGDPKMALDH1A1MEN1
SCHEMBL27880566 0.68 CDK5 (0.41) PKMALDH1A1CDK5CDK5R1CCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951244-A2 CALCILYTIC COMPOUNDS SmithKline Beecham Corporation (US) 2008-08-06 EP disclosed
WO-2007062370-A2 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-05-31 WO disclosed