SCHEMBL5147520

SCHEMBL5147520

CC1(C)NC(=O)N(CCNc2ncc(Br)c(-c3cc(CCO[Si](C)(C)C(C)(C)C)c(Cc4ccc(F)cc4)s3)n2)C1=O

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PLA2G7 Q13093 1/20 0.35
ALDH1A1 P00352 1/20 0.33
GRM2 Q14416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2974790 0.89
SCHEMBL5147508 0.86 PLA2G7 (0.34) PLA2G7ALDH1A1GRM2
SCHEMBL5145980 0.85 MAPK8 (0.34) PLA2G7ALDH1A1GRM2
SCHEMBL5148389 0.84 CA1 (0.35) PLA2G7ALDH1A1GRM2
SCHEMBL5147316 0.79 PLA2G7 (0.39) PLA2G7ALDH1A1GRM2
SCHEMBL5148399 0.79 PLA2G7 (0.39) PLA2G7ALDH1A1GRM2
SCHEMBL2980215 0.77
SCHEMBL2980503 0.76
SCHEMBL2971299 0.74
SCHEMBL5147336 0.74 PLA2G7 (0.35) PLA2G7ALDH1A1GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831207-A1 AMINOPYRIMIDINE COMPOUNDS AND METHODS OF USE Amgen Inc. (US) 2007-09-12 EP disclosed
WO-2006066172-A1 AMINOPYRIMIDINE COMPOUNDS AND METHODS OF USE AMGEN, INC. (US) 2006-06-22 WO disclosed