SCHEMBL5148362

SCHEMBL5148362

CC1(C)NC(=O)N(CCNc2nccc(-c3cc4cnccc4s3)n2)C1=O

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 1/20 0.39
CLK1 P49759 1/20 0.39
IKBKB O14920 7/20 0.39
CHUK O15111 5/20 0.37
IKBKG Q9Y6K9 5/20 0.37
CYP2A6 P11509 2/20 0.36
TGFBR1 P36897 9/20 0.36
MAPK14 Q16539 6/20 0.36
MAPK3 P27361 1/20 0.34
MAPK1 P28482 1/20 0.34
TGFB2 P61812 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5147360 0.87 CYP2A6 (0.35) CDK2CLK1CYP2A6TGFBR1MAPK14
SCHEMBL5147363 0.86 IKBKB (0.36) CDK2CLK1IKBKBCHUKIKBKG
SCHEMBL2989813 0.86 IKBKB (0.38) CDK2CLK1IKBKBCHUKIKBKG
SCHEMBL5147421 0.84 IKBKB (0.37) CDK2CLK1IKBKBCHUKIKBKG
SCHEMBL5147509 0.84 ALDH1A1 (0.38) CDK2CLK1IKBKBCHUKIKBKG
SCHEMBL5179013 0.82 ALDH1A1 (0.42) CDK2CLK1MAPK3MAPK1
SCHEMBL5147312 0.82 IKBKB (0.42) CDK2CLK1IKBKBMAPK1
SCHEMBL5147457 0.81 ALDH1A1 (0.40) CDK2CLK1MAPK3MAPK1
SCHEMBL5149101 0.81 RAF1 (0.37) TGFBR1MAPK14
SCHEMBL5147468 0.80 SMN1; SMN2 (0.40) CDK2CLK1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831207-A1 AMINOPYRIMIDINE COMPOUNDS AND METHODS OF USE Amgen Inc. (US) 2007-09-12 EP disclosed
WO-2006066172-A1 AMINOPYRIMIDINE COMPOUNDS AND METHODS OF USE AMGEN, INC. (US) 2006-06-22 WO disclosed