SCHEMBL5149573

SCHEMBL5149573

O=C1CSC(c2cccc(Cl)c2)N1CCc1ccccc1

nearest known ligand 0.76

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.64
POLB P06746 2/20 0.56
KMT2A Q03164 2/20 0.56
LMNA P02545 6/20 0.54
HPGD P15428 3/20 0.54
ALDH1A1 P00352 5/20 0.54
SMN1; SMN2 Q16637 4/20 0.53
KCNA5 P22460 1/20 0.52
MEN1 O00255 1/20 0.51
CACNA1B Q00975 1/20 0.51
HTT P42858 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
MAPT P10636 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5151414 0.83 ACHE (0.56) ACHEHPGDALDH1A1SMN1; SMN2KCNA5
SCHEMBL7254757 0.81 ACHE (0.71) ACHEPOLBNPSR1MAPT
SCHEMBL5152739 0.81 ACHE (0.58) ACHESMN1; SMN2CACNA1BNPSR1MAPT
SCHEMBL5152862 0.80 CACNA1B (0.74) POLBKMT2ALMNAHPGDALDH1A1
SCHEMBL5152821 0.80 CACNA1B (0.53) POLBKMT2ALMNAHPGDALDH1A1
SCHEMBL5156195 0.80 ACHE (0.65) ACHEPOLBNPSR1MAPT
SCHEMBL5151573 0.79 MAPT (0.67) ACHEPOLBKMT2AALDH1A1MEN1
SCHEMBL5152730 0.79 ACHE (0.71) ACHEPOLBNPSR1MAPT
SCHEMBL5156337 0.78 ACHE (0.63) ACHEPOLBKMT2A
SCHEMBL7250239 0.78 ACHE (0.66) ACHELMNAALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7223754-B2 Thiazolidinone, oxazolidinone, and imidazolone derivatives for treating lower urinary tract and related disorders DYNOGEN PHARMACEUTICALS, INC. (US) 2007-05-29 US disclosed
US-20070066597-A1 Thiazolidinone, oxazolidinone, and imidazolone derivatives for treating lower urinary tract and related disorders DYNOGEN PHARMACEUTICALS, INC. (US) 2007-03-22 US disclosed
US-20050148587-A1 Thiazolidinone, oxazolidinone, and imidazolone derivatives for treating lower urinary tract and related disorders DYNOGEN PHARMACEUTICALS, INC. (US) 2005-07-07 US disclosed
US-20050113421-A1 Thiazolidinone, oxazolidinone, and imidazolone derivatives for treating non-inflammatory gastrointestinal tract disorders DYNOGEN PHARMACEUTICALS, INC. (US) 2005-05-26 US disclosed
WO-2004017965-A1 1,3-THIAZOLIN-4-ONES AS THERAPEUTIC COMPOUNDS IN THE TREATMENT OF PAIN IONIX PHARMACEUTICALS LIMITED (GB) 2004-03-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050113421-A1 Thiazolidinone, oxazolidinone, and imidazolone derivatives for treating non-inflammatory gastrointestinal tract disorders TRPV2, RYR2, VDAC2 ACHE 3357/4885POLB 4811/4885KMT2A 4084/4885
US-20070066597-A1 Thiazolidinone, oxazolidinone, and imidazolone derivatives for treating lower urinary tract and related disorders RYR2, CACNB2, CACNA1I ACHE 3322/4885POLB 4735/4885KMT2A 3401/4885
US-20050148587-A1 Thiazolidinone, oxazolidinone, and imidazolone derivatives for treating lower urinary tract and related disorders RYR2, CACNB2, CACNA1I ACHE 3322/4885POLB 4735/4885KMT2A 3401/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.