SCHEMBL5155945

SCHEMBL5155945

CN(C)C1(Cc2ccc(Cl)cc2)CCC(NC(=O)COc2ccc(Cl)cc2)CC1.O=C(CCCOc1ccccc1)NC1CCC(c2ccccc2)(N2CCCCC2)CC1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ATF4 P18848 3/20 0.42
POLB P06746 1/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
HRH3 Q9Y5N1 2/20 0.39
USP2 O75604 1/20 0.39
ADIPOR2 Q86V24 1/20 0.39
ADIPOR1 Q96A54 1/20 0.39
ALDH1A1 P00352 2/20 0.39
LMNA P02545 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MCHR1 Q99705 1/20 0.38
RAB9A P51151 1/20 0.38
FAAH O00519 1/20 0.37
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2986952 0.85 MEN1 (0.47) ATF4MEN1KMT2ALMNARAB9A
SCHEMBL2976705 0.83 MEN1 (0.52) MEN1KMT2ASMN1; SMN2RAB9A
SCHEMBL2987483 0.81 ATF4 (0.61) ATF4POLBMEN1KMT2AUSP2
SCHEMBL2978761 0.80 ATF4 (0.65) ATF4POLBMEN1KMT2AALDH1A1
SCHEMBL2987110 0.79 MEN1 (0.51) POLBMEN1KMT2ASMN1; SMN2RAB9A
SCHEMBL2987816 0.77 MEN1 (0.47) MEN1KMT2ALMNARAB9A
SCHEMBL5159146 0.77 MEN1 (0.45) POLBMEN1KMT2AHRH3LMNA
SCHEMBL2977860 0.77 ATF4 (0.60) ATF4POLBMEN1KMT2ALMNA
SCHEMBL2985500 0.76 ATF4 (0.57) ATF4POLBMEN1KMT2AUSP2
SCHEMBL2982759 0.76 ATF4 (0.57) ATF4POLBMEN1KMT2AUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007536322-A 2007-12-13 JP claimed
EP-1747191-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES WITH A CHAIN EXTENSION Grünenthal GmbH (DE) 2007-01-31 EP claimed
WO-2005110975-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES WITH A CHAIN EXTENSION Grünenthal GmbH (DE) 2005-11-24 WO claimed