SCHEMBL5159146

SCHEMBL5159146

COCCOCC(=O)NC1CCC(Cc2ccc(C)cc2)(N(C)C)CC1.O=C(CCCOc1ccccc1)NC1CCC(Cc2ccccc2)(N2CCCCC2)CC1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
POLB P06746 1/20 0.37
RAB9A P51151 2/20 0.36
MAPT P10636 1/20 0.35
NPC1 O15118 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
EPHX2 P34913 1/20 0.34
LMNA P02545 1/20 0.34
BRD4 O60885 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
EPHX1 P07099 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2972836 0.83 MEN1 (0.50) MEN1KMT2APOLBRAB9AMAPT
SCHEMBL2981453 0.80 RAB9A (0.39) MEN1KMT2APOLBRAB9ANPC1
SCHEMBL2985450 0.79 OPRM1 (0.47) MEN1KMT2APOLBEPHX2HPGD
SCHEMBL2987110 0.79 MEN1 (0.51) MEN1KMT2APOLBRAB9AMAPT
SCHEMBL5155945 0.77 ATF4 (0.42) MEN1KMT2APOLBRAB9AHRH3
SCHEMBL2985459 0.77 POLB (0.59) MEN1KMT2APOLBRAB9ALMNA
SCHEMBL2983320 0.77 POLB (0.59) MEN1KMT2APOLBRAB9ALMNA
SCHEMBL2987472 0.76 NPSR1 (0.48) MEN1KMT2APOLBRAB9AMAPT
SCHEMBL2985703 0.76 MEN1 (0.59) MEN1KMT2ARAB9AMAPTNPC1
SCHEMBL2986952 0.75 MEN1 (0.47) MEN1KMT2ARAB9ANPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007536322-A 2007-12-13 JP claimed
EP-1747191-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES WITH A CHAIN EXTENSION Grünenthal GmbH (DE) 2007-01-31 EP claimed
WO-2005110975-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES WITH A CHAIN EXTENSION Grünenthal GmbH (DE) 2005-11-24 WO claimed