SCHEMBL5158397

SCHEMBL5158397

COc1ccc(-c2ncc(OC(=O)O)nc2-c2ccc(OC)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.54
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 3/20 0.46
LMNA P02545 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CHEK1 O14757 1/20 0.43
PTGS2 P35354 2/20 0.43
PTGDR2 Q9Y5Y4 2/20 0.43
KMT2A Q03164 2/20 0.42
RXFP1 Q9HBX9 1/20 0.41
EGLN1 Q9GZT9 1/20 0.41
HPGD P15428 1/20 0.41
MAPT P10636 2/20 0.41
GAA P10253 1/20 0.41
MEN1 O00255 1/20 0.40
PTGES O14684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5163847 0.83 CNR1 (0.49) CNR1ALDH1A1KDM4EHPGDGAA
SCHEMBL5160102 0.82 CNR1 (0.67) CNR1ALDH1A1KDM4ELMNANPSR1
SCHEMBL4455131 0.79 CNR1 (0.67) CNR1ALDH1A1KDM4ELMNANPSR1
SCHEMBL5163182 0.77 CNR1 (0.69) CNR1LMNAMAPT
SCHEMBL6454010 0.75 CNR1 (0.62) CNR1ALDH1A1KDM4ELMNANPSR1
SCHEMBL9695575 0.75 CNR1 (0.66) CNR1ALDH1A1KDM4ELMNAKMT2A
SCHEMBL9695458 0.73 THRB (0.51) CNR1ALDH1A1KDM4ELMNANPSR1
SCHEMBL9695460 0.73 THRB (0.51) CNR1ALDH1A1KDM4ELMNANPSR1
SCHEMBL10508434 0.73 ALDH1A1 (0.51) CNR1ALDH1A1KDM4ELMNANPSR1
SCHEMBL6223461 0.71 ESR2 (0.56) ALDH1A1LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1458690-B1 5,6-DIARYL-PYRAZINE-2-AMIDE DERIVATIVES AS CB1 ANTAGONISTS ASTRAZENECA AB (SE) 2007-02-21 EP claimed