SCHEMBL5158451

SCHEMBL5158451

CN(C)C1(Cc2ccc(Cl)cc2)CCC(NC(=O)CCC(=O)NC2CCc3ccccc32)CC1.CN(C)C1(Cc2ccc(Cl)cc2)CCC(NC(=O)CCC(=O)NCc2cccc(Br)c2)CC1.CN(C)C1(Cc2cccc(Cl)c2)CCC(NC(=O)CCC(=O)NC2CCc3ccccc32)CC1.Cc1cccc(CC2(N(C)C)CCC(NC(=O)CCC(=O)NCC(C)c3ccc(Cl)cc3)CC2)c1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 3/20 0.35
CCR2 P41597 3/20 0.33
NR1H4 Q96RI1 2/20 0.33
TRPV1 Q8NER1 1/20 0.33
POLB P06746 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
TP53 P04637 1/20 0.31
MAPT P10636 1/20 0.31
THRB P10828 1/20 0.31
SSTR1 P30872 1/20 0.31
SSTR4 P31391 1/20 0.31
BCL2L11 O43521 1/20 0.31
BCL2 P10415 1/20 0.31
MCL1 Q07820 1/20 0.31
KCNA5 P22460 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5159882 0.95 EPHX2 (0.36) DHODHCCR2NR1H4TRPV1
SCHEMBL4083007 0.83 DHODH (0.45) DHODHMEN1KMT2ATHRBNPSR1
SCHEMBL206128 0.82 SSTR1 (0.39) CCR2NR1H4MEN1KMT2ATHRB
SCHEMBL206834 0.80 DHODH (0.48) DHODHPOLBMEN1KMT2ATHRB
SCHEMBL206685 0.80 EPHX2 (0.43) POLBKMT2ATP53MAPTTHRB
SCHEMBL206533 0.80 CYP2C9 (0.42) CCR2NR1H4POLBKMT2ATHRB
SCHEMBL205814 0.80 LMNA (0.44) DHODHPOLBMEN1KMT2ATP53
SCHEMBL207581 0.79 POLB (0.46) NR1H4POLBKMT2ATP53MAPT
SCHEMBL206643 0.79 SSTR4 (0.43) NR1H4MEN1KMT2ASSTR1SSTR4
SCHEMBL207293 0.78 DHODH (0.48) DHODHPOLBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2007-01-24 EP disclosed
WO-2005110974-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2005-11-24 WO disclosed