SCHEMBL5325810

SCHEMBL5325810

COc1ccccc1-c1ccc2c(c1CN)[N]C(=O)C(=O)N2

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 4/20 0.45
CHEK1 O14757 1/20 0.43
NPC1 O15118 1/20 0.38
STK10 O94804 7/20 0.37
SLK Q9H2G2 7/20 0.37
HSD17B10 Q99714 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
GSK3B P49841 3/20 0.36
KDM4E B2RXH2 1/20 0.35
GPR55 Q9Y2T6 1/20 0.35
CREBBP Q92793 1/20 0.35
PRKCB P05771 1/20 0.35
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5158690 0.88 DPP4 (0.46) DPP4CHEK1STK10SLKHSD17B10
SCHEMBL1996958 0.69 DPP4 (0.46) DPP4HSD17B10ALDH1A1GAAKDM4E
SCHEMBL3149112 0.68 DPP4 (0.45) DPP4CHEK1NPC1HSD17B10ALDH1A1
SCHEMBL1993654 0.68 DPP4 (0.45) DPP4CHEK1NPC1ALDH1A1KDM4E
SCHEMBL3149462 0.65 DPP4 (0.57) DPP4HSD17B10ALDH1A1GSK3B
SCHEMBL6867119 0.65 TAAR1 (0.55) DPP4HSD17B10ALDH1A1GAA
SCHEMBL18170650 0.63 ADORA2A (0.54) CHEK1STK10SLKALDH1A1GSK3B
SCHEMBL4139350 0.62 IL6 (0.39) CHEK1STK10SLKHSD17B10ALDH1A1
SCHEMBL23611757 0.62 HSD17B10 (0.66) NPC1HSD17B10ALDH1A1GAAGSK3B
SCHEMBL3143679 0.62 DPP4 (1.00) DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007112347-A1 DIPEPTIDYL PEPTIDASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-10-04 WO claimed
WO-2007112347-A1 DIPEPTIDYL PEPTIDASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-10-04 WO disclosed