SCHEMBL5158738

SCHEMBL5158738

CCCN(C)C(=O)c1cnc(Cl)c(C(=O)O)c1.CCCN(C)C(=O)c1cnc(Cl)c(C(=O)OC)c1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 2/20 0.38
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 3/20 0.35
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KMT2A Q03164 2/20 0.34
DRD3 P35462 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
NAMPT P43490 2/20 0.34
GALK1 P51570 1/20 0.33
BCHE P06276 2/20 0.33
ACHE P22303 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
TSHR P16473 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3855168 0.95 ALDH1A1 (0.38) HCAR3KDM4EALDH1A1LMNAKMT2A
SCHEMBL3853097 0.92 HCAR3 (0.43) HCAR3KDM4EALDH1A1LMNAKMT2A
SCHEMBL28848352 0.78 KDM4E (0.46) HCAR3KDM4EALDH1A1MAPK1L3MBTL1
SCHEMBL3520084 0.75 MAPK1 (0.47) KDM4EALDH1A1LMNAMAPK1L3MBTL1
SCHEMBL3860560 0.73 ATM (0.51) KDM4EALDH1A1LMNAKMT2ANAMPT
SCHEMBL15391827 0.72 CYP2C9 (0.56) KDM4EALDH1A1LMNAMAPK1L3MBTL1
SCHEMBL15712178 0.70 MAPK1 (0.39) KDM4EALDH1A1MAPK1L3MBTL1TSHR
SCHEMBL3849724 0.70 PDE4A (0.42) KDM4EALDH1A1LMNAL3MBTL1KMT2A
SCHEMBL15391826 0.69 CYP2C9 (0.56) KDM4EALDH1A1LMNAMAPK1KMT2A
SCHEMBL3517645 0.69 HCAR2 (0.48) KDM4EALDH1A1LMNAKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740575-A2 PYRROLIDINE DERIVATIVES USEFUL AS BACE INHIBITORS ELI LILLY AND COMPANY (US) 2007-01-10 EP disclosed
WO-2005108358-A2 PYRROLIDINE DERIVATIVES USEFUL AS BACE INHIBITORS ELI LILLY AND COMPANY (US) 2005-11-17 WO disclosed