SCHEMBL5159399

SCHEMBL5159399

CCCN(C)c1cc(C(=O)O)cc(S(C)(=O)=O)n1.COC(=O)c1cc(Cl)nc(S(C)(=O)=O)c1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 2/20 0.38
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 3/20 0.33
CYP1A2 P05177 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GPR119 Q8TDV5 3/20 0.32
LMNA P02545 1/20 0.32
CNR1 P21554 1/20 0.32
MAPT P10636 2/20 0.31
BACE1 P56817 1/20 0.31
L3MBTL1 Q9Y468 2/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
PPARG P37231 1/20 0.31
PPARA Q07869 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3858500 0.89 LMNA (0.38) HCAR3ALDH1A1KDM4ECYP1A2TSHR
SCHEMBL3860981 0.86 HCAR3 (0.49) HCAR3ALDH1A1TSHRSMN1; SMN2CNR1
SCHEMBL3857572 0.83 ALDH1A1 (0.43) HCAR3ALDH1A1KDM4ECYP1A2TSHR
SCHEMBL3856420 0.80 ALDH1A1 (0.46) ALDH1A1KDM4ECYP1A2TSHRCYP2C19
SCHEMBL3350040 0.77 ALDH1A1 (0.41) ALDH1A1KDM4ELMNACNR1MAPT
SCHEMBL3855487 0.76 KDM4E (0.39) HCAR3ALDH1A1KDM4ECYP1A2TSHR
SCHEMBL1816292 0.74 ALDH1A1 (0.40) ALDH1A1KDM4ECYP1A2TSHRCYP2C19
SCHEMBL1579300 0.74 ALDH1A1 (0.43) ALDH1A1KDM4ELMNAL3MBTL1
SCHEMBL3854447 0.74 POLB (0.39) HCAR3ALDH1A1KDM4ECYP1A2TSHR
SCHEMBL3720398 0.73 ALDH1A1 (0.42) ALDH1A1KDM4ELMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740573-A1 AMIDES AS BACE INHIBITORS ELI LILLY AND COMPANY (US) 2007-01-10 EP disclosed
WO-2005108391-A1 AMIDES AS BACE INHIBITORS ELI LILLY AND COMPANY (US) 2005-11-17 WO disclosed