SCHEMBL5160899

SCHEMBL5160899

CC(C(=O)O)C(=O)c1ccncn1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.47
GRM4 Q14833 3/20 0.40
FAAH O00519 1/20 0.38
BRD4 O60885 1/20 0.38
BRPF1 P55201 1/20 0.38
CTNNB1 P35222 2/20 0.38
WNT3A P56704 2/20 0.38
TBXA2R P21731 4/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
GSK3B P49841 2/20 0.34
GSK3A P49840 1/20 0.34
CHRM2 P08172 1/20 0.33
GRM5 P41594 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8016097 0.83 P2RX7 (0.52) P2RX7GRM4FAAHBRD4BRPF1
SCHEMBL5161602 0.83 P2RX7 (0.45) P2RX7GRM4FAAHBRD4BRPF1
SCHEMBL4411674 0.79 P2RX7 (0.49) P2RX7GRM4FAAHBRD4BRPF1
SCHEMBL3567261 0.79 P2RX7 (0.45) P2RX7GRM4FAAHBRD4BRPF1
SCHEMBL5558104 0.79 P2RX7 (0.47) P2RX7GRM4FAAHBRD4BRPF1
SCHEMBL13729034 0.78 POLB (0.44) P2RX7GRM4TBXA2RCYP1A2CYP3A4
SCHEMBL13827559 0.77 P2RX7 (0.50) P2RX7GRM4FAAHBRD4BRPF1
SCHEMBL5160643 0.76 GSK3B (0.59) ALDH1A1GSK3BLMNA
SCHEMBL29587616 0.74
SCHEMBL37469 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1340746-B1 Process for the reduction of 3-heteroaryl-3-oxo-propanoic acid derivatives SALTIGO GMBH (DE) 2007-02-28 EP disclosed
EP-1340746-A1 Process for the reduction of 3-heteroaryl-3-oxo-propanoic acid derivatives BAYER AG (DE) 2003-09-03 EP disclosed