SCHEMBL5161602

SCHEMBL5161602

CC(C)C(C(=O)O)C(=O)c1ccncn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.45
GRM4 Q14833 2/20 0.38
FAAH O00519 1/20 0.37
BRD4 O60885 1/20 0.36
BRPF1 P55201 1/20 0.36
CTNNB1 P35222 2/20 0.36
WNT3A P56704 2/20 0.36
TBXA2R P21731 4/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
GSK3B P49841 2/20 0.33
GSK3A P49840 1/20 0.33
XIAP P98170 1/20 0.32
BIRC2 Q13490 1/20 0.32
IP6K1 Q92551 1/20 0.32
IP6K3 Q96PC2 1/20 0.32
IP6K2 Q9UHH9 1/20 0.32
CHRM2 P08172 1/20 0.32
GRM5 P41594 1/20 0.32
SIGMAR1 Q99720 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5160899 0.83 P2RX7 (0.47) P2RX7GRM4FAAHBRD4BRPF1
SCHEMBL8016097 0.80 P2RX7 (0.52) P2RX7GRM4FAAHBRD4BRPF1
SCHEMBL5163592 0.78 GSK3B (0.56) CYP1A2CYP3A4GSK3BLMNA
SCHEMBL4411674 0.77 P2RX7 (0.49) P2RX7GRM4FAAHBRD4BRPF1
SCHEMBL5558104 0.76 P2RX7 (0.47) P2RX7GRM4FAAHBRD4BRPF1
SCHEMBL13729034 0.75 POLB (0.44) P2RX7GRM4TBXA2RCYP1A2CYP3A4
SCHEMBL5162688 0.75 NAPRT (0.48) CYP1A2CYP3A4LMNA
SCHEMBL5160371 0.75 FAAH (0.45) P2RX7FAAHCTNNB1WNT3ATBXA2R
SCHEMBL13827559 0.75 P2RX7 (0.50) P2RX7GRM4FAAHBRD4BRPF1
Bromide SCHEMBL10349040 0.74 P2RX7 (0.57) P2RX7GRM4FAAHCTNNB1WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1340746-B1 Process for the reduction of 3-heteroaryl-3-oxo-propanoic acid derivatives SALTIGO GMBH (DE) 2007-02-28 EP disclosed
EP-1340746-A1 Process for the reduction of 3-heteroaryl-3-oxo-propanoic acid derivatives BAYER AG (DE) 2003-09-03 EP disclosed