SCHEMBL5160982

SCHEMBL5160982

COC(=O)CCc1cnc(N2CCC[C@H]2COC(C)C(=O)Cc2cc(Cl)c(NC(=O)c3coc4ccccc34)cc2F)s1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 9/20 0.39
ITGB1 P05556 8/20 0.39
GPBAR1 Q8TDU6 1/20 0.33
TP53 P04637 3/20 0.32
TDP1 Q9NUW8 1/20 0.32
THRB P10828 1/20 0.31
EGFR P00533 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
MAP4K1 Q92918 2/20 0.30
NTRK1 P04629 1/20 0.30
CHRM3 P20309 1/20 0.30
PIM2 Q9P1W9 1/20 0.30
ACKR3 P25106 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5414719 0.90 ITGA4 (0.40) ITGA4ITGB1GPBAR1TP53TDP1
SCHEMBL5410475 0.85 ITGB1 (0.40) ITGA4ITGB1TP53TDP1THRB
SCHEMBL5160221 0.84 ITGB1 (0.45) ITGA4ITGB1TP53TDP1EGFR
SCHEMBL5160791 0.84 ITGA4 (0.40) ITGA4ITGB1GPBAR1TP53THRB
SCHEMBL5160984 0.83 ITGB1 (0.38) ITGA4ITGB1GPBAR1TP53TDP1
SCHEMBL5175632 0.81 ITGB1 (0.37) ITGA4ITGB1TP53TDP1THRB
SCHEMBL5158240 0.80 ITGB1 (0.48) ITGA4ITGB1TP53TDP1THRB
SCHEMBL5160816 0.79 ITGB1 (0.40) ITGA4ITGB1TP53TDP1MAP4K1
SCHEMBL5176215 0.79 ITGB1 (0.52) ITGA4ITGB1ALDH1A1MAP4K1NTRK1
SCHEMBL5422528 0.79 ITGB1 (0.46) ITGA4ITGB1TP53TDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070232601-A1 Vla-4 Inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2007-10-04 US disclosed
EP-1757602-A1 VLA-4 INHIBITOR DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2007-02-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070232601-A1 Vla-4 Inhibitor VCAM1, ITGB4, ITGA4 ITGA4 3/4885ITGB1 9/4885GPBAR1 1464/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.