SCHEMBL5161747

SCHEMBL5161747

COC(=O)[C@@H](N)Cc1ccc(-c2cn(C)c(=O)n(C)c2=O)c(C)c1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 7/20 0.55
ITGA4 P13612 7/20 0.55
ITGB7 P26010 3/20 0.55
ALDH1A1 P00352 1/20 0.41
PTGS2 P35354 1/20 0.35
ERN1 O75460 1/20 0.34
HSD17B10 Q99714 2/20 0.34
GAA P10253 1/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
SLC7A5 Q01650 2/20 0.33
POLB P06746 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
TP53 P04637 1/20 0.31
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27511850 0.88 ITGB1 (0.61) ITGB1ITGA4ITGB7PTGS2HSD17B10
SCHEMBL27511849 0.88 ITGB1 (0.61) ITGB1ITGA4ITGB7PTGS2HSD17B10
SCHEMBL5163064 0.84 ITGA4 (0.39) ITGB1ITGA4ITGB7ALDH1A1PTGS2
Hydrochloric Acid SCHEMBL5165900 0.83 ALDH1A1 (0.41) ITGB1ITGA4ITGB7ALDH1A1PTGS2
SCHEMBL5162201 0.83 ITGB1 (0.55) ITGB1ITGA4ITGB7ALDH1A1PTGS2
SCHEMBL5162949 0.79 ITGA4 (0.59) ITGB1ITGA4ITGB7ALDH1A1TSHR
SCHEMBL5159923 0.78 ITGA4 (0.84) ITGB1ITGA4ITGB7
SCHEMBL27488188 0.76 DPP4 (0.42) ITGA4ITGB7ALDH1A1PTGS2
SCHEMBL27488187 0.76 DPP4 (0.42) ITGA4ITGB7ALDH1A1PTGS2
SCHEMBL22996698 0.75 ITGB1 (0.45) ITGB1ITGA4ITGB7ALDH1A1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1237878-B1 4-PYRIMIDINYL-N-ACYL-L-PHENYLALANINES HOFFMANN LA ROCHE (CH) 2007-03-21 EP disclosed
EP-1237878-A2 4-PYRIMIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2002-09-11 EP disclosed
US-6380387-B1 ANTIINFLAMMATORY AGENTS, ANTIASTHMATICS HOFFMANN-LA ROCHE INC. 2002-04-30 US disclosed
WO-2001042225-A2 4-PYRIMIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2001-06-14 WO disclosed